Fragment-Based Anti-inflammatory Agent Design and Target Identification: Discovery of AF-45 as an IRAK4 Inhibitor to Treat Ulcerative Colitis and Acute Lung Injury
基于片段的抗炎剂设计和靶标识别:发现 AF-45 作为 IRAK4 抑制剂可治疗溃疡性结肠炎和急性肺损伤
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.4c00202
Yu Zou, Xiemin Wang, Pan Chen, Zhiwei Zheng, Xiaobo Li, Zhichao Chen, Mi Guo, Ying Zhou, Chenhui Sun, Ran Wang, Wufu Zhu, Pengwu Zheng, Won-Jea Cho, Young-Chang Cho, Guang Liang, Qidong Tang