日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

LYMTACs:chimeric small molecules repurpose lysosomal membrane proteins for target protein relocalization and degradation.

LYMTACs:嵌合小分子可重新利用溶酶体膜蛋白,实现靶蛋白的重新定位和降解

Nalawansha Dhanusha A, Mazis Georgios, Husemoen Gitte, Ashton Kate S, Deng Weixian, Wurz Ryan P, Tran Anh T, Lanman Brian A, Xie Jiansong, Guenette Robert G, Li Shiqian, Smith Christopher E, Archunan Suresh, Agnihotram Manoj K, Sadhukhan Arghya, Kapoor Rajiv, Wilde Chris, Koirala Sajjan, De Sousa E Melo Felipe, Potts Patrick Ryan

Structural Elucidation and Absolute Stereochemistry for Pharma Compounds Using MicroED

利用微型电子衍射技术进行药物化合物的结构解析和绝对立体化学测定

de Moraes, Lygia Silva; Burch, Jessica E; Delgadillo, David A; Rodriguez, Isabel Hernandez; Mai, Huanghao; Smith, Austin G; Caille, Seb; Walker, Shawn D; Wurz, Ryan P; Cee, Victor J; Rodriguez, Jose A; Gostovic, Dan; Quasdorf, Kyle; Nelson, Hosea M

Photoinduced, Copper-Catalyzed Decarboxylative C-N Coupling to Generate Protected Amines: An Alternative to the Curtius Rearrangement

光诱导铜催化脱羧CN偶联生成保护胺:一种替代库尔提乌斯重排的方法

Zhao, Wei; Wurz, Ryan P; Peters, Jonas C; Fu, Gregory C

Discovery and Optimization of Macrocyclic Quinoxaline-pyrrolo-dihydropiperidinones as Potent Pim-1/2 Kinase Inhibitors

发现和优化大环喹喔啉-吡咯并二氢哌啶酮类化合物作为强效Pim-1/2激酶抑制剂

Cee, Victor J; Chavez, Frank Jr; Herberich, Bradley; Lanman, Brian A; Pettus, Liping H; Reed, Anthony B; Wu, Bin; Wurz, Ryan P; Andrews, Kristin L; Chen, Jie; Hickman, Dean; Laszlo, Jimmy 3rd; Lee, Matthew R; Guerrero, Nadia; Mattson, Bethany K; Nguyen, Yen; Mohr, Christopher; Rex, Karen; Sastri, Christine E; Wang, Paul; Wu, Qiong; Wu, Tian; Xu, Yang; Zhou, Yihong; Winston, Jeffrey T; Lipford, J Russell; Tasker, Andrew S; Wang, Hui-Ling

Oxopyrido[2,3-d]pyrimidines as Covalent L858R/T790M Mutant Selective Epidermal Growth Factor Receptor (EGFR) Inhibitors

氧代吡啶并[2,3-d]嘧啶类化合物作为共价L858R/T790M突变选择性表皮生长因子受体(EGFR)抑制剂

Wurz, Ryan P; Pettus, Liping H; Ashton, Kate; Brown, James; Chen, Jian Jeffrey; Herberich, Brad; Hong, Fang-Tsao; Hu-Harrington, Essa; Nguyen, Tom; St Jean, David J Jr; Tadesse, Seifu; Bauer, David; Kubryk, Michele; Zhan, Jinghui; Cooke, Keegan; Mitchell, Petia; Andrews, Kristin L; Hsieh, Faye; Hickman, Dean; Kalyanaraman, Nataraj; Wu, Tian; Reid, Darren L; Lobenhofer, Edward K; Andrews, Dina A; Everds, Nancy; Guzman, Roberto; Parsons, Andrew T; Hedley, Simon J; Tedrow, Jason; Thiel, Oliver R; Potter, Matthew; Radinsky, Robert; Beltran, Pedro J; Tasker, Andrew S