日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Targeting PLK1 potentiates the antitumor efficacy of EGFR-TKIs through inhibiting the JAK1/STAT3 pathway

靶向PLK1可通过抑制JAK1/STAT3通路增强EGFR-TKIs的抗肿瘤疗效。

Li, Cheng; Shi, Shangxuan; Li, Long; Wang, Yafang; Yao, Mingyue; Yu, Chengcheng; Yu, Chuwei; Xie, Chengying

IHCH9033, a novel class I HDAC inhibitor, synergizes with FLT3 inhibitor and rescues quizartinib resistance in FLT3-ITD AML via enhancing DNA damage response

IHCH9033 是一种新型 I 类 HDAC 抑制剂,可与 FLT3 抑制剂产生协同作用,并通过增强 DNA 损伤反应来逆转 FLT3-ITD AML 中的 quizartinib 耐药性。

Yao, Mingyue; Yan, Wenzhong; Wang, Yafang; Zhao, Yu; Xu, Xiaowei; Chen, Yujun; Yu, Chengcheng; Li, Yingnian; Jiang, Hualiang; Shen, Jie; Cheng, Jianjun; Xie, Chengying

Synthesis and Anticancer Activity Evaluation of Novel Carborane-Containing Isoflavonoid Analogues

新型含碳硼烷异黄酮类似物的合成及抗癌活性评价

Zhang, Yirong; Yu, Chuwei; Wang, Linyuan; Zhou, Lina; Li, Chaofan; Yuan, Changxian; Sun, Nan; Hao, Guanxiang; Ma, Chenyang; Lin, Yuzhe; Li, Hongjing; Hong, Jiali; Zhao, Jinhua; Lou, Kaiyan; Zhang, Rui; Xie, Chengying; Wang, Sinan

Unraveling the CDK9/PP2A/ERK Network in Transcriptional Pause Release and Complement Activation in KRAS-mutant Cancers

揭示KRAS突变癌症中CDK9/PP2A/ERK网络在转录暂停解除和补体激活中的作用

Wang, Yafang; Xu, Lansong; Ling, Lijun; Yao, Mingyue; Shi, Shangxuan; Yu, Chengcheng; Li, Yingnian; Shen, Jie; Jiang, Hualiang; Xie, Chengying

IRAK1 deficiency potentiates the efficacy of radiotherapy in repressing cervical cancer development

IRAK1 缺乏可增强放射治疗抑制宫颈癌发展的功效

Wenjuan Chen, Xingyun Xie, Chengying Liu, Jingrong Liao, Yuting Wei, Rongrong Wu, Jinsheng Hong

In vivo flow cytometry reveals a circadian rhythm of circulating tumor cells

体内流式细胞术揭示循环肿瘤细胞的昼夜节律

Zhu, Xi; Suo, Yuanzhen; Fu, Yuting; Zhang, Fuli; Ding, Nan; Pang, Kai; Xie, Chengying; Weng, Xiaofu; Tian, Meilu; He, Hao; Wei, Xunbin

Pharmacologic characterization of fluzoparib, a novel poly(ADP-ribose) polymerase inhibitor undergoing clinical trials

氟唑帕尼(一种正在进行临床试验的新型聚(ADP-核糖)聚合酶抑制剂)的药理学特征

Wang, Lei; Yang, Changyong; Xie, Chengying; Jiang, Jiahua; Gao, Mingzhao; Fu, Li; Li, Yun; Bao, Xubin; Fu, Haoyu; Lou, Liguang

Preclinical characterization of SHR6390, a novel CDK 4/6 inhibitor, in vitro and in human tumor xenograft models.

在体外和人类肿瘤异种移植模型中对新型 CDK 4/6 抑制剂 SHR6390 进行临床前表征

Long Fei, He Ye, Fu Haoyu, Li Yun, Bao Xubin, Wang Quanren, Wang Yigang, Xie Chengying, Lou Liguang

Preclinical characterization of anlotinib, a highly potent and selective vascular endothelial growth factor receptor-2 inhibitor

安罗替尼(一种高效且选择性的血管内皮生长因子受体-2抑制剂)的临床前特性研究

Xie, Chengying; Wan, Xiaozhe; Quan, Haitian; Zheng, Mingyue; Fu, Li; Li, Yun; Lou, Liguang

Puquitinib, a novel orally available PI3Kδ inhibitor, exhibits potent antitumor efficacy against acute myeloid leukemia

Puquitinib 是一种新型口服 PI3Kδ 抑制剂,对急性髓系白血病具有强大的抗肿瘤疗效。

Xie, Chengying; He, Ye; Zhen, Mingyue; Wang, Yulan; Xu, Yongping; Lou, Liguang