日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of Niclosamide Analogs with Potent Mitochondrial Uncoupling Activity and Reduced Mitochondrial Inhibition-Associated Toxicity

发现具有强效线粒体解偶联活性和降低线粒体抑制相关毒性的尼克酰胺类似物

Jiang, Haowen; Macorano, Alessio; Xing, Enming; Jedoui, Mohamed; Mohammed, Shabber; Lee, Vanessa; Cheng, Jeffrey; McDonough, Lain; Cheng, Xiaolin; Ye, Jiangbin; Li, Pui Kai

TopMT-GAN: a 3D topology-driven generative model for efficient and diverse structure-based ligand design

TopMT-GAN:一种基于三维拓扑结构的高效多样化配体设计生成模型

Wang, Shen; Lin, Tong; Peng, Tianyi; Xing, Enming; Chen, Sijie; Kara, Levent Burak; Cheng, Xiaolin

Valine-Niclosamide for Treatment of Androgen Receptor Splice Variant-Positive Hepatocellular Carcinoma.

缬氨酸-尼克酰胺用于治疗雄激素受体剪接变异体阳性肝细胞癌

Hoelzen Emma J, Radomska Hanna S, Kulp Samuel K, Adeluola Adeoluwa A, Granchie Lauren A, Cheng Jeffrey, Dauki Anees M, Campbell Moray J, Mohammed Shabber, Xing Enming, Hai Min, Fukuda Mayu, Cheng Xiaolin, Phelps Mitch A, Li Pui-Kai, Coss Christopher C

Netupitant Exhibits Potent Activity on Mycobacterium tuberculosis Persisters

奈妥匹坦对结核分枝杆菌持续菌表现出强效活性

Eldesouky, Hassan E; Jones, Richard M; Mohammed, Shabber; Xing, Enming; Li, Pui-Kai; Sherman, David R

Leveraging Sequence Purification for Accurate Prediction of Multiple Conformational States with AlphaFold2

利用序列纯化技术,通过 AlphaFold2 精确预测多种构象状态

Xing, Enming; Zhang, Junjie; Wang, Shen; Cheng, Xiaolin

The pH gradient contributes to persistence in Mycobacterium tuberculosis

pH梯度有助于结核分枝杆菌的持续存在

Sherman, David; Eldesouky, Hassan; Adams, Kristin; Brache, Justin; Aguila, Laarni; Garcia, Mariana; Xing, Enming; Li, Pui-Kai

LX1 Dual Targets AR Variants and AKR1C3 in Advanced Prostate Cancer Therapy.

LX1 双靶点 AR 变异体和 AKR1C3 在晚期前列腺癌治疗中的应用

Ning Shu, Armstrong Cameron M, Xing Enming, Leslie Amy R, Gao Richard Y, Sharifi Masuda, Schaaf Zachary A, Lou Wei, Han Xiangrui, Xu Desiree H, Yang Rui, Cheng Jeffrey, Mohammed Shabber, Mitsiades Nicholas, Liu Chengfei, Lombard Alan P, Wu Chun-Yi, Cheng Xiaolin, Li Pui-Kai, Gao Allen C

Anti-friction gold-based stretchable electronics enabled by interfacial diffusion-induced cohesion

通过界面扩散诱导的内聚力实现抗摩擦金基可拉伸电子器件

Jie Cao, Xusheng Liu, Jie Qiu, Zhifei Yue, Yang Li, Qian Xu, Yan Chen, Jiewen Chen, Hongfei Cheng, Guozhong Xing, Enming Song, Ming Wang, Qi Liu, Ming Liu1

BET Bromodomain Inhibitors: Novel Design Strategies and Therapeutic Applications

BET溴结构域抑制剂:新型设计策略和治疗应用

To, Kenneth K W; Xing, Enming; Larue, Ross C; Li, Pui-Kai

Cycloruthenated Self-Assembly with Metabolic Inhibition to Efficiently Overcome Multidrug Resistance in Cancers

环钌化自组装结合代谢抑制可有效克服癌症多药耐药性

Li, Jia; Zeng, Leli; Wang, Zheng; Chen, Hengxing; Fang, Shuo; Wang, Jinquan; Cai, Chao-Yun; Xing, Enming; Liao, Xinxing; Li, Zhi-Wei; Ashby, Charles R Jr; Chen, Zhe-Sheng; Chao, Hui; Pan, Yihang