Enhancing intracellular accumulation and target engagement of PROTACs with reversible covalent chemistry
利用可逆共价化学增强 PROTAC 的细胞内积累和靶向结合
期刊:Nature Communications
影响因子:14.7
doi:10.1038/s41467-020-17997-6
Wen-Hao Guo #, Xiaoli Qi #, Xin Yu, Yang Liu, Chan-I Chung, Fang Bai, Xingcheng Lin, Dong Lu, Lingfei Wang, Jianwei Chen, Lynn Hsiao Su, Krystle J Nomie, Feng Li, Meng C Wang, Xiaokun Shu, José N Onuchic, Jennifer A Woyach, Michael L Wang, Jin Wang