日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-Based Development of Ultra-Broad-Spectrum 3C-Like Protease Inhibitors

基于结构的超广谱3C样蛋白酶抑制剂的开发

Su, Haixia; Nie, Tianqing; Chen, Guofeng; Xiong, Muya; Zhang, Yumin; Wu, Guoqing; You, Mengyuan; Xie, Hang; He, Jian; Xiong, Yanchao; Hu, Hangchen; Zhao, Wenfeng; Li, Minjun; Xiao, Gengfu; Zhang, Leike; Xu, Yechun

De novo design of protein condensation inhibitors by targeting an allosteric site of cGAS.

通过靶向 cGAS 的变构位点,从头设计蛋白质缩合抑制剂

Zhao Wenfeng, Chen Guofeng, He Jian, Shen Xiaofang, Xiong Muya, Xiong Liwei, Qi Zhihao, Xie Hang, Li Wanchen, Li Jiameng, Dou Huixia, Hu Hangchen, Su Haixia, Shao Qiang, Li Minjun, Sun Hongbin, Xu Yechun

Structure-based design of potent and selective inhibitors targeting RIPK3 for eliminating on-target toxicity in vitro.

基于结构的高效选择性RIPK3抑制剂设计,可消除体外靶向毒性

Su Haixia, Chen Guofeng, Xie Hang, Li Wanchen, Xiong Muya, He Jian, Hu Hangchen, Zhao Wenfeng, Shao Qiang, Li Minjun, Zhao Qiang, Xu Yechun

Dynamic Cap-Mediated Substrate Access and Potent Inhibitor Design of Monkeypox Virus I7L Protease

猴痘病毒I7L蛋白酶的动态帽介导底物进入和强效抑制剂设计

Su, Haixia; Wu, Guoqing; Xiong, Muya; Wang, Yuhang; Cao, Junyuan; You, Mengyuan; Xiang, Yingchun; Nie, Tianqing; Li, Minjun; Xiao, Gengfu; Zhang, Leike; Shao, Qiang; Xu, Yechun

Benzbromarone interferes with the interaction between Hsp90 and Aha1 by interacting with both of them.

苯溴马隆通过与 Hsp90 和 Aha1 相互作用,干扰二者之间的相互作用

Zhong Yan, Shi Li, Xu Zhuo, Gao Jing, Ma Qingyu, Gao Tianqi, Tang Junying, Xiong Muya, Xu Yechun, Dai Huixiong, Zhou Hu, Zhang Naixia, Zhou Chen

Multi-omics for COVID-19: driving development of therapeutics and vaccines

新冠病毒多组学:推动治疗药物和疫苗的研发

Guo, Mengyu; Xiong, Muya; Peng, Jinying; Guan, Tong; Su, Haixia; Huang, Yanyi; Yang, Cai-Guang; Li, Yang; Boraschi, Diana; Pillaiyar, Thanigaimalai; Wang, Guanbo; Yi, Chengqi; Xu, Yechun; Chen, Chunying

Unraveling the catalytic mechanism of SARS-CoV-2 papain-like protease with allosteric modulation of C270 mutation using multiscale computational approaches

利用多尺度计算方法揭示SARS-CoV-2木瓜蛋白酶样蛋白酶的催化机制及其对C270突变的变构调节作用

Shao, Qiang; Xiong, Muya; Li, Jiameng; Hu, Hangchen; Su, Haixia; Xu, Yechun

Allosteric Regulation of Hsp90α's Activity by Small Molecules Targeting the Middle Domain of the Chaperone

小分子靶向分子伴侣中间结构域对Hsp90α活性的变构调节

Zhou, Chen; Zhang, Chi; Zhu, Hongwen; Liu, Zhijun; Su, Haixia; Zhang, Xianglei; Chen, Tingting; Zhong, Yan; Hu, Huifang; Xiong, Muya; Zhou, Hu; Xu, Yechun; Zhang, Ao; Zhang, Naixia