日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-Based Development of Ultra-Broad-Spectrum 3C-Like Protease Inhibitors

基于结构的超广谱3C样蛋白酶抑制剂的开发

Su, Haixia; Nie, Tianqing; Chen, Guofeng; Xiong, Muya; Zhang, Yumin; Wu, Guoqing; You, Mengyuan; Xie, Hang; He, Jian; Xiong, Yanchao; Hu, Hangchen; Zhao, Wenfeng; Li, Minjun; Xiao, Gengfu; Zhang, Leike; Xu, Yechun

Fusion Strategy of DNA-Encoded Libraries Drives Discovery of Allosteric Inhibitors of SARS-CoV‑2 RdRp

DNA编码文库的融合策略推动了SARS-CoV-2 RNA依赖性RNA聚合酶(RdRp)变构抑制剂的发现。

Li, Linjie; Wang, Xudong; Ding, Peiqi; Shen, Xuanjing; Hu, Hangchen; Wang, Xiaoxi; Jin, Rui; Wu, Xinyuan; Zhang, Yiwei; Lu, Weiwei; Yue, Jinfeng; Xu, H Eric; Yin, Wanchao; Xu, Yechun; Lu, Xiaojie

Author Correction: PPIA dictates NRF2 stability to promote lung cancer progression

作者更正:PPIA 决定 NRF2 的稳定性以促进肺癌进展

Lu, Weiqiang; Cui, Jiayan; Wang, Wanyan; Hu, Qian; Xue, Yun; Liu, Xi; Gong, Ting; Lu, Yiping; Ma, Hui; Yang, Xinyu; Feng, Bo; Wang, Qi; Zhang, Naixia; Xu, Yechun; Liu, Mingyao; Nussinov, Ruth; Cheng, Feixiong; Ji, Hongbin; Huang, Jin

De novo design of protein condensation inhibitors by targeting an allosteric site of cGAS.

通过靶向 cGAS 的变构位点,从头设计蛋白质缩合抑制剂

Zhao Wenfeng, Chen Guofeng, He Jian, Shen Xiaofang, Xiong Muya, Xiong Liwei, Qi Zhihao, Xie Hang, Li Wanchen, Li Jiameng, Dou Huixia, Hu Hangchen, Su Haixia, Shao Qiang, Li Minjun, Sun Hongbin, Xu Yechun

Structure-based design of potent and selective inhibitors targeting RIPK3 for eliminating on-target toxicity in vitro.

基于结构的高效选择性RIPK3抑制剂设计,可消除体外靶向毒性

Su Haixia, Chen Guofeng, Xie Hang, Li Wanchen, Xiong Muya, He Jian, Hu Hangchen, Zhao Wenfeng, Shao Qiang, Li Minjun, Zhao Qiang, Xu Yechun

Dynamic Cap-Mediated Substrate Access and Potent Inhibitor Design of Monkeypox Virus I7L Protease

猴痘病毒I7L蛋白酶的动态帽介导底物进入和强效抑制剂设计

Su, Haixia; Wu, Guoqing; Xiong, Muya; Wang, Yuhang; Cao, Junyuan; You, Mengyuan; Xiang, Yingchun; Nie, Tianqing; Li, Minjun; Xiao, Gengfu; Zhang, Leike; Shao, Qiang; Xu, Yechun

Benzbromarone interferes with the interaction between Hsp90 and Aha1 by interacting with both of them.

苯溴马隆通过与 Hsp90 和 Aha1 相互作用,干扰二者之间的相互作用

Zhong Yan, Shi Li, Xu Zhuo, Gao Jing, Ma Qingyu, Gao Tianqi, Tang Junying, Xiong Muya, Xu Yechun, Dai Huixiong, Zhou Hu, Zhang Naixia, Zhou Chen

Unveiling the Genetic Diversity and Population Structure of the Endangered Fern Angiopteris fokiensis Through Genome Survey and Genomic SSR Markers

通过基因组调查和基因组SSR标记揭示濒危蕨类植物福建海蕨的遗传多样性和种群结构

Zhou, Yiwei; Tan, Jianjun; Huang, Lishan; Luo, Yanyu; Huang, Shaoli; Ye, Yuanjun; Xu, Yechun

Oral Simnotrelvir for Adult Patients with Mild-to-Moderate Covid-19

口服西诺替韦治疗轻度至中度新冠肺炎成人患者

Cao, Bin; Wang, Yeming; Lu, Hongzhou; Huang, Chaolin; Yang, Yumei; Shang, Lianhan; Chen, Zhu; Jiang, Rongmeng; Liu, Yihe; Lin, Ling; Peng, Ping; Wang, Fuxiang; Gong, Fengyun; Hu, Honglin; Cheng, Cong; Yao, Xiangyang; Ye, Xianwei; Zhou, Hourong; Shen, Yinzhong; Liu, Chenfan; Wang, Chunying; Yi, Zhennan; Hu, Bijie; Xu, Jiuyang; Gu, Xiaoying; Shen, Jingshan; Xu, Yechun; Zhang, Leike; Fan, Jia; Tang, Renhong; Wang, Chen

Covalent DNA-Encoded Library Workflow Drives Discovery of SARS-CoV-2 Nonstructural Protein Inhibitors

共价DNA编码文库工作流程推动SARS-CoV-2非结构蛋白抑制剂的发现

Wang, Xudong; Xiong, Liwei; Zhu, Ying; Liu, Sixiu; Zhao, Wenfeng; Wu, Xinyuan; Seydimemet, Mengnisa; Li, Linjie; Ding, Peiqi; Lin, Xian; Liu, Jiaxiang; Wang, Xuan; Duan, Zhiqiang; Lu, Weiwei; Suo, Yanrui; Cui, Mengqing; Yue, Jinfeng; Jin, Rui; Zheng, Mingyue; Xu, Yechun; Mei, Lianghe; Hu, Hangchen; Lu, Xiaojie