日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Development of dual aptamers-functionalized c-MET PROTAC degraders for targeted therapy of osteosarcoma

双适体功能化的 c-MET PROTAC 降解剂的开发用于骨肉瘤的靶向治疗

Xuekun Fu, Jie Huang, Xinxin Chen, Duoli Xie, Hongzhen Chen, Zhijian Liang, Zhuqian Wang, Yiying Liang, Aiping Lu, Chao Liang

A Sponge-like Polysaccharide from Pine Pollen: Structural Features and Therapeutic Potential in DNCB-Induced Atopic Dermatitis Models

松花粉海绵状多糖:结构特征及其在DNCB诱导的特应性皮炎模型中的治疗潜力

Qiu, Zhuoya; Zhang, Mengru; Du, Haitao; Wang, Yi; Shao, Xuekun; Fu, Jialei; Wang, Ping; Wang, Cheng

Gut microbial metabolite targets HDAC3-FOXK1-interferon axis in fibroblast-like synoviocytes to ameliorate rheumatoid arthritis

肠道微生物代谢物靶向成纤维细胞样滑膜细胞中的 HDAC3-FOXK1-干扰素轴以改善类风湿性关节炎

Hongzhen Chen #, Xuekun Fu #, Xiaohao Wu #, Junyi Zhao, Fang Qiu, Zhenghong Wang, Zhuqian Wang, Xinxin Chen, Duoli Xie, Jie Huang, Junyu Fan, Xu Yang, Yi Song, Jie Li, Dongyi He, Guozhi Xiao, Aiping Lu, Chao Liang

Repurposing AS1411 for constructing ANM-PROTACs

重新利用 AS1411 构建 ANM-PROTAC

Xuekun Fu, Jin Li, Xinxin Chen, Hongzhen Chen, Zhuqian Wang, Fang Qiu, Duoli Xie, Jie Huang, Siran Yue, Chunhao Cao, Yiying Liang, Aiping Lu, Chao Liang

Poly (ADP-ribose) polymerase 1 (PARP1) inhibition promotes pulmonary metastasis of osteosarcoma by boosting ezrin phosphorylation

聚(ADP-核糖)聚合酶 1(PARP1)抑制通过促进埃兹蛋白磷酸化促进骨肉瘤肺转移

Fangfei Li, Xiaoqiu Wu, Xuekun Fu, Jin Liu, Wangze Song, Gary Guishan Xiao, Aiping Lu, Ge Zhang

Andrographolide prevents bone loss via targeting estrogen-related receptor-α-regulated metabolic adaption of osteoclastogenesis

穿心莲内酯通过靶向雌激素相关受体 α 调节破骨细胞生成的代谢适应来防止骨质流失

Tongling Huang, Xuekun Fu, Na Wang, Meng Yang, Minyi Zhang, Binxu Wang, Tianke Chen, Sidra Majaz, Huaiyu Wang, Chi-Wai Wong, Jinsong Liu, Min Guan

Kindlin-2 mediates mechanotransduction in bone by regulating expression of Sclerostin in osteocytes

Kindlin-2 通过调节骨细胞中 Sclerostin 的表达来介导骨骼中的机械转导

Lei Qin #, Xuekun Fu #, Jing Ma, Manxia Lin, Peijun Zhang, Yishu Wang, Qinnan Yan, Chu Tao, Wen Liu, Bin Tang, Di Chen, Xiaochun Bai, Huiling Cao, Guozhi Xiao

ALKAL1 gene silencing prevents colorectal cancer progression via suppressing Sonic Hedgehog (SHH) signaling pathway

ALKAL1 基因沉默通过抑制 Sonic Hedgehog (SHH) 信号通路阻止结直肠癌进展

Shasha Chen, Bin Wang, Xuekun Fu, Yanfang Liang, Xingxing Chai, Ziyu Ye, Ronggang Li, Yaoming He, Gang Kong, Jiachun Lian, Xiangyong Li, Ting Chen, Xin Zhang, Xianxiu Qiu, Xudong Tang, Keyuan Zhou, Bihua Lin, Jincheng Zeng

Kindlin-2 regulates skeletal homeostasis by modulating PTH1R in mice

Kindlin-2 通过调节小鼠的 PTH1R 来调节骨骼稳态

Xuekun Fu, Bo Zhou, Qinnan Yan, Chu Tao, Lei Qin, Xiaohao Wu, Sixiong Lin, Sheng Chen, Yumei Lai, Xuenong Zou, Zengwu Shao, Meiqing Wang, Di Chen, Wenfei Jin, Youqiang Song, Huiling Cao, Ge Zhang, Guozhi Xiao2

LIM domain proteins Pinch1/2 regulate chondrogenesis and bone mass in mice

LIM 结构域蛋白 Pinch1/2 调节小鼠的软骨形成和骨量

Yiming Lei #, Xuekun Fu #, Pengyu Li #, Sixiong Lin, Qinnan Yan, Yumei Lai, Xin Liu, Yishu Wang, Xiaochun Bai, Chuanju Liu, Di Chen, Xuenong Zou, Xu Cao, Huiling Cao, Guozhi Xiao