日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Rationally designed Fe-cyclopentadienone with unique orientations for efficient asymmetric hydrogenation of acylsilanes

合理设计的具有独特取向的铁-环戊二烯酮可高效不对称氢化酰基硅烷

Xie, Chaochao; Yao, Bo-Xuan; Law, Kwok-Chung; Zhang, Xumu; Ni, Shao-Fei; Tan, Xuefeng

Anti-SARS-CoV-2 prodrug ATV006 has broad-spectrum antiviral activity against human and animal coronaviruses

抗SARS-CoV-2前药ATV006对人类和动物冠状病毒具有广谱抗病毒活性

Xu, Tiefeng; Li, Kun; Huang, Siyao; Ivanov, Konstantin I; Yang, Sidi; Ji, Yanxi; Zhang, Hanwei; Wu, Wenbin; He, Ye; Zeng, Qiang; Cong, Feng; Zhou, Qifan; Li, Yingjun; Pan, Jian; Zhao, Jincun; Li, Chunmei; Zhang, Xumu; Cao, Liu; Guo, Deyin

Preclinical characterization and anti-RSV efficacy of an oral C-nucleoside derivative

口服C-核苷衍生物的临床前表征及其抗RSV疗效

Chen, Yuanguang; Liu, Yongqing; Li, Guanguan; Peng, Chao; Liang, Dizhen; Yang, Sidi; Zheng, Peisen; Li, Shuo; Guo, Deyin; Zhou, Qifan; Zhang, Xumu

Broad-Spectrum Antiviral Activity of the Orally Bioavailable Antiviral ATV014 Against Multiple Coronaviruses

口服生物利用度高的抗病毒药物ATV014对多种冠状病毒具有广谱抗病毒活性

Yang, Sidi; Li, Kun; Zhou, Qifan; Zhang, Xumu; Guo, Deyin

Gram-scale synthesis of (+)-elacestrant streamlined by iridium-catalyzed dynamic kinetic asymmetric hydrogenation of α-substituted tetralones

利用铱催化的α-取代四氢萘酮动态动力学不对称氢化反应,简化了(+)-elacestrant的克级合成。

Zong, Yan; Zou, Xiaomei; Zhang, Shaoke; Chen, Gen-Qiang; Zhang, Xumu

Efficacy and safety of SHEN26, a novel oral small molecular RdRp inhibitor for COVID-19 treatment: a multicenter, randomized, double-blinded, placebo-controlled, phase II clinical trial

新型口服小分子RdRp抑制剂SHEN26治疗COVID-19的疗效和安全性:一项多中心、随机、双盲、安慰剂对照的II期临床试验

Bai, Jiangtao; Asakawa, Tetsuya; Yuan, Wenfang; Lin, Yuanlong; Ju, Hao; Xu, Dandan; Yang, Mingming; Li, Shuo; Li, Guanguan; Guo, Deyin; Lu, Hongzhou; Zhang, Xumu

Chemo-, regio- and enantioselective hydroformylation of trisubstituted cyclopropenes: access to chiral quaternary cyclopropanes

三取代环丙烯的化学选择性、区域选择性和对映选择性氢甲酰化:手性季碳环丙烷的合成

Li, Shuailong; Zhang, Dequan; Purushothaman, Aiswarya; Lv, Hui; Shilpa, Shilpa; Sunoj, Raghavan B; Li, Xiuxiu; Zhang, Xumu

Robust, scalable, and highly selective spirocyclic catalysts for industrial hydroformylation and isomerization-hydroformylation

用于工业氢甲酰化和异构化-氢甲酰化的稳健、可扩展且高选择性的螺环催化剂

Zong, Yan; Zhang, Runtong; Ma, Baode; Peng, Jianghua; Wu, Chao; Zou, Xiaomei; Qian, Yu; Chen, Gen-Qiang; Zhang, Xumu

Facile access to chiral γ-butyrolactones via rhodium-catalysed asymmetric hydrogenation of γ-butenolides and γ-hydroxybutenolides

通过铑催化的γ-丁烯内酯和γ-羟基丁烯内酯的不对称氢化反应,简便地合成手性γ-丁内酯

Zhou, Yuxuan; Guo, Siyuan; Huang, Qiyuan; Lang, Qiwei; Chen, Gen-Qiang; Zhang, Xumu

Highly enantioselective synthesis of both tetrahydroquinoxalines and dihydroquinoxalinones via Rh-thiourea catalyzed asymmetric hydrogenation

通过铑-硫脲催化的不对称氢化反应,高对映选择性地合成四氢喹喔啉和二氢喹喔啉酮。

Xu, Ana; Li, Chaoyi; Huang, Junrong; Pang, Heng; Zhao, Chengyao; Song, Lijuan; You, Hengzhi; Zhang, Xumu; Chen, Fen-Er