Synthesis and biological evaluation of 4-(4-aminophenyl)-6-methylisoxazolo[3,4-b] pyridin-3-amine covalent inhibitors as potential agents for the treatment of acute myeloid leukemia
4-(4-氨基苯基)-6-甲基异恶唑并[3,4-b]吡啶-3-胺共价抑制剂的合成及作为治疗急性髓系白血病的潜在药物的生物学评价
期刊:Bioorganic & Medicinal Chemistry
影响因子:3.3
doi:10.1016/j.bmc.2022.116937
Ji-Bo Kang, Lu Chen, Xue-Jiao Leng, Jing-Jing Wang, Yang Cheng, Shi-Han Wu, Yi-Yuan Ma, Li-Jin Yang, Yu-Hao Cao, Xiao Yang, Zhen-Jiang Tong, Jia-Zhen Wu, Yi-Bo Wang, Hai Zhou, Jia-Chuan Liu, Ning Ding, Wei-Chen Dai, Yan-Cheng Yu, Xin Xue, Shan-Liang Sun, Xiao-Bin Dai, Liang Chang, Xiao-Long Wang, Ni