Discovery of a novel thiophene carboxamide analogue as a highly potent and selective sphingomyelin synthase 2 inhibitor for dry eye disease therapy.
发现一种新型噻吩甲酰胺类似物,可作为高效选择性的鞘磷脂合成酶 2 抑制剂用于治疗干眼症
期刊:Acta Pharmaceutica Sinica B
影响因子:14.6
doi:10.1016/j.apsb.2024.10.005
Yang Jintong, Lu Yiteng, Hu Kexin, Zhang Xinchen, Wang Wei, Ye Deyong, Mo Mingguang, Xiao Xin, Wan Xichen, Wu Yuqing, Zhang Shuxian, Huang He, Qu Zhibei, Hu Yimin, Cao Yu, Hong Jiaxu, Zhou Lu