日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery and development of a new oxazolidinone with reduced toxicity for the treatment of tuberculosis

发现和开发一种毒性降低的新型噁唑烷酮类药物用于治疗结核病

Crowley, Brendan M; Boshoff, Helena I; Boving, Aidan; Tan, Vee Y; Zhu, Jianghai; Hoyt, Forrest; Miller, Randy R; Ehrhart, Julie; Boyce, Christopher W; Young, Katherine; Nantermet, Philippe G; Su, Jing; Yang, Lihu; Painter, Ronald E; Corcoran, Emily B; Hoar, Jason L; Oh, Sangmi; Holtzman, David L; Levi, Micha; Anderson, Aparna; Otieno, Monicah A; Zimmerman, Matthew; Kaya, Firat; Massoudi, Lisa M; Ramey, Michelle E; Bauman, Allison A; Lenaerts, Anne J; Roberston, Gregory T; Dartois, Véronique; Wells, Charles D; Barry, Clifton E 3rd; Olsen, David B

Linking High-Throughput Screens to Identify MoAs and Novel Inhibitors of Mycobacterium tuberculosis Dihydrofolate Reductase

利用高通量筛选鉴定结核分枝杆菌二氢叶酸还原酶的作用机制和新型抑制剂

Santa Maria, John P Jr; Park, Yumi; Yang, Lihu; Murgolo, Nicholas; Altman, Michael D; Zuck, Paul; Adam, Greg; Chamberlin, Chad; Saradjian, Peter; Dandliker, Peter; Boshoff, Helena I M; Barry, Clifton E 3rd; Garlisi, Charles; Olsen, David B; Young, Katherine; Glick, Meir; Nickbarg, Elliott; Kutchukian, Peter S

Discovery of MK-7145, an Oral Small Molecule ROMK Inhibitor for the Treatment of Hypertension and Heart Failure

发现MK-7145,一种用于治疗高血压和心力衰竭的口服小分子ROMK抑制剂

Tang, Haifeng; Zhu, Yuping; Teumelsan, Nardos; Walsh, Shawn P; Shahripour, Aurash; Priest, Birgit T; Swensen, Andrew M; Felix, John P; Brochu, Richard M; Bailey, Timothy; Thomas-Fowlkes, Brande; Pai, Lee-Yuh; Hampton, Caryn; Corona, Aaron; Hernandez, Melba; Metzger, Joseph; Forrest, Michael; Zhou, Xiaoyan; Owens, Karen; Tong, Vincent; Parmee, Emma; Roy, Sophie; Kaczorowski, Gregory J; Yang, Lihu; Alonso-Galicia, Magdalena; Garcia, Maria L; Pasternak, Alexander

Stimulation of Glucose-Dependent Insulin Secretion by a Potent, Selective sst3 Antagonist

强效选择性 sst3 拮抗剂刺激葡萄糖依赖性胰岛素分泌

Pasternak, Alexander; Feng, Zhe; de Jesus, Reynalda; Ye, Zhixiong; He, Shuwen; Dobbelaar, Peter; Bradley, Scott A; Chicchi, Gary G; Tsao, Kwei-Lan; Trusca, Dorina; Eiermann, George J; Li, Cai; Feng, Yue; Wu, Margaret; Shao, Qing; Zhang, Bei B; Nargund, Ravi; Mills, Sander G; Howard, Andrew D; Yang, Lihu; Zhou, Yun-Ping

The Discovery of MK-4256, a Potent SSTR3 Antagonist as a Potential Treatment of Type 2 Diabetes

MK-4256是一种强效的SSTR3拮抗剂,其作为2型糖尿病潜在治疗方法的发现

He, Shuwen; Ye, Zhixiong; Truong, Quang; Shah, Shrenik; Du, Wu; Guo, Liangqin; Dobbelaar, Peter H; Lai, Zhong; Liu, Jian; Jian, Tianying; Qi, Hongbo; Bakshi, Raman K; Hong, Qingmei; Dellureficio, James; Pasternak, Alexander; Feng, Zhe; deJesus, Reynalda; Yang, Lihu; Reibarkh, Mikhail; Bradley, Scott A; Holmes, Mark A; Ball, Richard G; Ruck, Rebecca T; Huffman, Mark A; Wong, Frederick; Samuel, Koppara; Reddy, Vijay B; Mitelman, Stan; Tong, Sharon X; Chicchi, Gary G; Tsao, Kwei-Lan; Trusca, Dorina; Wu, Margaret; Shao, Qing; Trujillo, Maria E; Eiermann, George J; Li, Cai; Zhang, Bei B; Howard, Andrew D; Zhou, Yun-Ping; Nargund, Ravi P; Hagmann, William K

Dual targeting of CCR2 and CX3CR1 in an arterial injury model of vascular inflammation.

在血管炎症的动脉损伤模型中,对 CCR2 和 CX3CR1 进行双重靶向治疗

Jerath Maya R, Liu Peng, Struthers Mary, Demartino Julie A, Peng Roche, Peterson Laurence B, Cumiskey Anne-Marie, Yang Lihu, Rojas Mauricio, Patel Dhavalkumar D, Fong Alan M