Discovery and Preclinical Evaluations of Potent, Selective, and Allosteric Covalent WRN Inhibitors with Improved PK Properties
发现并进行临床前评估高效、选择性强、具有改进药代动力学特性的变构共价WRN抑制剂
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.5c00787
Xu, Zhaobing; Xiao, Qi; Liu, Yong; Jiang, Wen; Liu, Lifei; Sun, Hongna; Yang, Xiulan; Lu, Zhuojian; Yan, Bocheng; Long, Hanxiong; Zhang, Xuejun