日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Targeting transcription in heart failure via CDK7/12/13 inhibition

通过抑制 CDK7/12/13 靶向心力衰竭中的转录

Austin Hsu #, Qiming Duan #, Daniel S Day #, Xin Luo, Sarah McMahon, Yu Huang, Zachary B Feldman, Zhen Jiang, Tinghu Zhang, Yanke Liang, Michael Alexanian, Arun Padmanabhan, Jonathan D Brown, Charles Y Lin, Nathanael S Gray, Richard A Young, Benoit G Bruneau, Saptarsi M Haldar

Mapping the Degradable Kinome Provides a Resource for Expedited Degrader Development

绘制可降解激酶组图谱为加速降解剂开发提供资源

Katherine A Donovan, Fleur M Ferguson, Jonathan W Bushman, Nicholas A Eleuteri, Debabrata Bhunia, SeongShick Ryu, Li Tan, Kun Shi, Hong Yue, Xiaoxi Liu, Dennis Dobrovolsky, Baishan Jiang, Jinhua Wang, Mingfeng Hao, Inchul You, Mingxing Teng, Yanke Liang, John Hatcher, Zhengnian Li, Theresa D Manz, B

A broad-spectrum antiviral molecule, QL47, selectively inhibits eukaryotic translation

广谱抗病毒分子 QL47 选择性抑制真核翻译

Mélissanne de Wispelaere, Margot Carocci, Dominique J Burri, William J Neidermyer Jr, Calla M Olson, Imme Roggenbach, Yanke Liang, Jinhua Wang, Sean P J Whelan, Nathanael S Gray, Priscilla L Yang

A kinase-independent role for CDK8 in BCR-ABL1+ leukemia

CDK8 在 BCR-ABL1+ 白血病中发挥激酶非依赖性作用

Ingeborg Menzl, Tinghu Zhang, Angelika Berger-Becvar, Reinhard Grausenburger, Gerwin Heller, Michaela Prchal-Murphy, Leo Edlinger, Vanessa M Knab, Iris Z Uras, Eva Grundschober, Karin Bauer, Mareike Roth, Anna Skucha, Yao Liu, John M Hatcher, Yanke Liang, Nicholas P Kwiatkowski, Daniela Fux, Andrea

Homolog-Selective Degradation as a Strategy to Probe the Function of CDK6 in AML

同源物选择性降解作为探究 CDK6 在 AML 中功能的策略

Matthias Brand, Baishan Jiang, Sophie Bauer, Katherine A Donovan, Yanke Liang, Eric S Wang, Radosław P Nowak, Jingting C Yuan, Tinghu Zhang, Nicholas Kwiatkowski, André C Müller, Eric S Fischer, Nathanael S Gray, Georg E Winter

Development of a Selective CDK7 Covalent Inhibitor Reveals Predominant Cell-Cycle Phenotype

选择性 CDK7 共价抑制剂的开发揭示了主要的细胞周期表型

Calla M Olson, Yanke Liang, Alan Leggett, Woojun D Park, Lianbo Li, Caitlin E Mills, Selma Z Elsarrag, Scott B Ficarro, Tinghu Zhang, Robert Düster, Matthias Geyer, Taebo Sim, Jarrod A Marto, Peter K Sorger, Ken D Westover, Charles Y Lin, Nicholas Kwiatkowski, Nathanael S Gray

Development of Dual and Selective Degraders of Cyclin-Dependent Kinases 4 and 6

细胞周期蛋白依赖性激酶 4 和 6 的双重和选择性降解剂的开发

Baishan Jiang, Eric S Wang, Katherine A Donovan, Yanke Liang, Eric S Fischer, Tinghu Zhang, Nathanael S Gray

Pharmacological perturbation of CDK9 using selective CDK9 inhibition or degradation

使用选择性 CDK9 抑制或降解对 CDK9 进行药理学干扰

Calla M Olson, Baishan Jiang, Michael A Erb, Yanke Liang, Zainab M Doctor, Zinan Zhang, Tinghu Zhang, Nicholas Kwiatkowski, Myriam Boukhali, Jennifer L Green, Wilhelm Haas, Tyzoon Nomanbhoy, Eric S Fischer, Richard A Young, James E Bradner, Georg E Winter, Nathanael S Gray

Targeting MYC dependency in ovarian cancer through inhibition of CDK7 and CDK12/13

通过抑制 CDK7 和 CDK12/13 靶向卵巢癌中的 MYC 依赖性

Mei Zeng, Nicholas P Kwiatkowski, Tinghu Zhang, Behnam Nabet, Mousheng Xu, Yanke Liang, Chunshan Quan, Jinhua Wang, Mingfeng Hao, Sangeetha Palakurthi, Shan Zhou, Qing Zeng, Paul T Kirschmeier, Khyati Meghani, Alan L Leggett, Jun Qi, Geoffrey I Shapiro, Joyce F Liu, Ursula A Matulonis, Charles Y Lin

A UV-Independent Topical Small-Molecule Approach for Melanin Production in Human Skin

一种不依赖紫外线的局部小分子方法,用于抑制人体皮肤黑色素的产生

Nisma Mujahid, Yanke Liang, Ryo Murakami, Hwan Geun Choi, Allison S Dobry, Jinhua Wang, Yusuke Suita, Qing Yu Weng, Jennifer Allouche, Lajos V Kemeny, Andrea L Hermann, Elisabeth M Roider, Nathanael S Gray, David E Fisher