日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Integrated Approach of Machine Learning and High-Throughput Screening to Identify Chemical Probe Candidates Targeting Aldehyde Dehydrogenases.

机器学习与高通量筛选相结合的方法来识别靶向醛脱氢酶的化学探针候选物。

Yasgar Adam, Jain Sankalp, Davies Marissa, Danchik Carina, Niehoff Taylor, Ran Jing, Rai Ganesha, Yang Shyh-Ming, Simeonov Anton, Zakharov Alexey V, Martinez Natalia J

Quantitative Bioactivity Signatures of Dietary Supplements and Natural Products

膳食补充剂和天然产物的定量生物活性特征

Yasgar, Adam; Bougie, Danielle; Eastman, Richard T; Huang, Ruili; Itkin, Misha; Kouznetsova, Jennifer; Lynch, Caitlin; McKnight, Crystal; Miller, Mitch; Ngan, Deborah K; Peryea, Tyler; Shah, Pranav; Shinn, Paul; Xia, Menghang; Xu, Xin; Zakharov, Alexey V; Simeonov, Anton

A platform of assays for the discovery of anti-Zika small-molecules with activity in a 3D-bioprinted outer-blood-retina model

用于发现对3D生物打印外血视网膜模型具有活性的抗寨卡小分子的检测平台

Dorjsuren, Dorjbal; Eastman, Richard T; Song, Min Jae; Yasgar, Adam; Chen, Yuchi; Bharti, Kapil; Zakharov, Alexey V; Jadhav, Ajit; Ferrer, Marc; Shi, Pei-Yong; Simeonov, Anton

The Tox21 10K Compound Library: Collaborative Chemistry Advancing Toxicology

Tox21 10K化合物库:协作化学推动毒理学发展

Richard, Ann M; Huang, Ruili; Waidyanatha, Suramya; Shinn, Paul; Collins, Bradley J; Thillainadarajah, Inthirany; Grulke, Christopher M; Williams, Antony J; Lougee, Ryan R; Judson, Richard S; Houck, Keith A; Shobair, Mahmoud; Yang, Chihae; Rathman, James F; Yasgar, Adam; Fitzpatrick, Suzanne C; Simeonov, Anton; Thomas, Russell S; Crofton, Kevin M; Paules, Richard S; Bucher, John R; Austin, Christopher P; Kavlock, Robert J; Tice, Raymond R

Optimization of High-Throughput Methyltransferase Assays for the Discovery of Small Molecule Inhibitors

优化高通量甲基转移酶检测方法以发现小分子抑制剂

Dong, Guangping; Yasgar, Adam; Peterson, Darrell L; Zakharov, Alexey; Talley, Daniel; Cheng, Ken Chih-Chien; Jadhav, Ajit; Simeonov, Anton; Huang, Rong

Canvass: A Crowd-Sourced, Natural-Product Screening Library for Exploring Biological Space

Canvass:一个用于探索生物空间的众包天然产物筛选库

Kearney, Sara E; Zahoránszky-Kőhalmi, Gergely; Brimacombe, Kyle R; Henderson, Mark J; Lynch, Caitlin; Zhao, Tongan; Wan, Kanny K; Itkin, Zina; Dillon, Christopher; Shen, Min; Cheff, Dorian M; Lee, Tobie D; Bougie, Danielle; Cheng, Ken; Coussens, Nathan P; Dorjsuren, Dorjbal; Eastman, Richard T; Huang, Ruili; Iannotti, Michael J; Karavadhi, Surendra; Klumpp-Thomas, Carleen; Roth, Jacob S; Sakamuru, Srilatha; Sun, Wei; Titus, Steven A; Yasgar, Adam; Zhang, Ya-Qin; Zhao, Jinghua; Andrade, Rodrigo B; Brown, M Kevin; Burns, Noah Z; Cha, Jin K; Mevers, Emily E; Clardy, Jon; Clement, Jason A; Crooks, Peter A; Cuny, Gregory D; Ganor, Jake; Moreno, Jesus; Morrill, Lucas A; Picazo, Elias; Susick, Robert B; Garg, Neil K; Goess, Brian C; Grossman, Robert B; Hughes, Chambers C; Johnston, Jeffrey N; Joullie, Madeleine M; Kinghorn, A Douglas; Kingston, David G I; Krische, Michael J; Kwon, Ohyun; Maimone, Thomas J; Majumdar, Susruta; Maloney, Katherine N; Mohamed, Enas; Murphy, Brian T; Nagorny, Pavel; Olson, David E; Overman, Larry E; Brown, Lauren E; Snyder, John K; Porco, John A Jr; Rivas, Fatima; Ross, Samir A; Sarpong, Richmond; Sharma, Indrajeet; Shaw, Jared T; Xu, Zhengren; Shen, Ben; Shi, Wei; Stephenson, Corey R J; Verano, Alyssa L; Tan, Derek S; Tang, Yi; Taylor, Richard E; Thomson, Regan J; Vosburg, David A; Wu, Jimmy; Wuest, William M; Zakarian, Armen; Zhang, Yufeng; Ren, Tianjing; Zuo, Zhong; Inglese, James; Michael, Sam; Simeonov, Anton; Zheng, Wei; Shinn, Paul; Jadhav, Ajit; Boxer, Matthew B; Hall, Matthew D; Xia, Menghang; Guha, Rajarshi; Rohde, Jason M

Corrigendum: A PHGDH inhibitor reveals coordination of serine synthesis and one-carbon unit fate

更正:PHGDH 抑制剂揭示了丝氨酸合成与一碳单元命运的协调性

Pacold, Michael E; Brimacombe, Kyle R; Chan, Sze Ham; Rohde, Jason M; Lewis, Caroline A; Swier, Lotteke J Y M; Possemato, Richard; Chen, Walter W; Sullivan, Lucas B; Fiske, Brian P; Cho, Steve; Freinkman, Elizaveta; Birsoy, Kıvanç; Abu, Monther-Remaileh; Shaul, Yoav D; Liu, Chieh Min; Zhou, Minerva; Koh, Min Jung; Chung, Haeyoon; Davidson, Shawn M; Luengo, Alba; Wang, Amy Q; Xu, Xin; Yasgar, Adam; Liu, Li; Rai, Ganesha; Westover, Kenneth D; Heiden, Matthew G Vander; Shen, Min; Gray, Nathanael S; Boxer, Matthew B; Sabatini, David M

Fluorescence polarization assays in high-throughput screening and drug discovery: a review

荧光偏振分析在高通量筛选和药物发现中的应用:综述

Hall, Matthew D; Yasgar, Adam; Peryea, Tyler; Braisted, John C; Jadhav, Ajit; Simeonov, Anton; Coussens, Nathan P

AlphaScreen-Based Assays: Ultra-High-Throughput Screening for Small-Molecule Inhibitors of Challenging Enzymes and Protein-Protein Interactions

基于AlphaScreen的检测方法:超高通量筛选难阻酶和蛋白质-蛋白质相互作用的小分子抑制剂

Yasgar, Adam; Jadhav, Ajit; Simeonov, Anton; Coussens, Nathan P

Current approaches for the discovery of drugs that deter substance and drug abuse

目前用于发现可抑制物质和药物滥用的药物的方法

Yasgar, Adam; Simeonov, Anton