日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of 7-Azanorbornane-Based Dual Agonists for the Delta and Kappa Opioid Receptors through an In Situ Screening Protocol

通过原位筛选方案发现基于 7-Azanorbornane 的 Delta 和 Kappa 阿片受体双重激动剂

Fumika Karaki, Taro Takamori, Koumei Kawakami, Sae Sakurai, Kyoko Hidaka, Kei Ishii, Tomoya Oki, Noriko Sato, Nao Atsumi, Karin Ashizawa, Ai Taguchi, Asuka Ura, Toko Naruse, Shigeto Hirayama, Miki Nonaka, Kanako Miyano, Yasuhito Uezono, Hideaki Fujii

The Steroidal Alkaloid Tomatidine and Tomatidine-Rich Tomato Leaf Extract Suppress the Human Gastric Cancer-Derived 85As2 Cells In Vitro and In Vivo via Modulation of Interferon-Stimulated Genes

类固醇生物碱番茄碱和富含番茄碱的番茄叶提取物通过调节干扰素刺激基因抑制人胃癌衍生的 85As2 细胞

Junya Fujimaki, Neo Sayama, Shigenobu Shiotani, Takanori Suzuki, Miki Nonaka, Yasuhito Uezono, Mamoru Oyabu, Yasutomi Kamei, Haruo Nukaya, Keiji Wakabayashi, Akihito Morita, Tomoki Sato, Shinji Miura

Novel Opioid Analgesics for the Development of Transdermal Opioid Patches That Possess Morphine-Like Pharmacological Profiles Rather Than Fentanyl: Possible Opioid Switching Alternatives Among Patch Formula

新型阿片类镇痛药,用于开发具有与吗啡类似药理学特性而非芬太尼的透皮阿片类贴剂:贴剂配方中可能的阿片类药物转换替代方案

Akane Komatsu, Kanako Miyano, Daisuke Nakayama, Yusuke Mizobuchi, Eiko Uezono, Kaori Ohshima, Yusuke Karasawa, Yui Kuroda, Miki Nonaka, Keisuke Yamaguchi, Masako Iseki, Yasuhito Uezono, Masakazu Hayashida

Peripherally administered cisplatin activates a parvocellular neuronal subtype expressing arginine vasopressin and enhanced green fluorescent protein in the paraventricular nucleus of a transgenic rat

外周给药顺铂可激活转基因大鼠室旁核中表达精氨酸加压素和增强型绿色荧光蛋白的细小细胞神经元亚型

Yasuki Akiyama, Mitsuhiro Yoshimura, Hiromichi Ueno, Kenya Sanada, Kentaro Tanaka, Satomi Sonoda, Haruki Nishimura, Kazuaki Nishimura, Yasuhito Motojima, Reiko Saito, Takashi Maruyama, Keiji Hirata, Yasuhito Uezono, Yoichi Ueta

Differential Metabolic Responses to Adipose Atrophy Associated with Cancer Cachexia and Caloric Restriction in Rats and the Effect of Rikkunshito in Cancer Cachexia

大鼠癌症恶病质和热量限制引起的脂肪萎缩的差异代谢反应以及六君子汤对癌症恶病质的影响

Yuka Sudo, Hiroki Otsuka, Ryota Miyakawa, Akifumi Goto, Yohei Kashiwase, Kiyoshi Terawaki, Kanako Miyano, Yuto Hirao, Kanari Taki, Ryoma Tagawa, Masaki Kobayashi, Naoyuki Okita, Yasuhito Uezono, Yoshikazu Higami

Leukemia inhibitory factor via the Toll-like receptor 5 signaling pathway involves aggravation of cachexia induced by human gastric cancer-derived 85As2 cells in rats

白血病抑制因子通过 Toll 样受体 5 信号通路加重大鼠人胃癌衍生 85As2 细胞诱发的恶病质

Kiyoshi Terawaki, Yohei Kashiwase, Miaki Uzu, Miki Nonaka, Yumi Sawada, Kanako Miyano, Yoshikazu Higami, Kazuyoshi Yanagihara, Masahiro Yamamoto, Yasuhito Uezono

Relief from neuropathic pain by blocking of the platelet-activating factor-pain loop

通过阻断血小板活化因子-疼痛环路缓解神经性疼痛

Hideo Shindou, Seiji Shiraishi, Suzumi M Tokuoka, Yoshikazu Takahashi, Takeshi Harayama, Takaya Abe, Kana Bando, Kanako Miyano, Yoshihiro Kita, Yasuhito Uezono, Takao Shimizu

Identification of Lysophosphatidic Acid Receptor 1 in Astroglial Cells as a Target for Glial Cell Line-derived Neurotrophic Factor Expression Induced by Antidepressants

鉴定星形胶质细胞中的溶血磷脂酸受体 1 作为抗抑郁药诱导的胶质细胞系衍生神经营养因子表达的靶点

Naoto Kajitani, Kanako Miyano, Mami Okada-Tsuchioka, Hiromi Abe, Kei Itagaki, Kazue Hisaoka-Nakashima, Norimitsu Morioka, Yasuhito Uezono, Minoru Takebayashi

Peripheral opioid antagonist enhances the effect of anti-tumor drug by blocking a cell growth-suppressive pathway in vivo

外周阿片类拮抗剂通过阻断体内细胞生长抑制通路增强抗肿瘤药物的作用

Masami Suzuki, Fumiko Chiwaki, Yumi Sawada, Maho Ashikawa, Kazuhiko Aoyagi, Takeshi Fujita, Kazuyoshi Yanagihara, Masayuki Komatsu, Minoru Narita, Tsutomu Suzuki, Hiroshi Nagase, Ryoji Kushima, Hiromi Sakamoto, Takeo Fukagawa, Hitoshi Katai, Hitoshi Nakagama, Teruhiko Yoshida, Yasuhito Uezono, Hirok