日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Design, synthesis and anti-breast cancer activity evaluation of 6,7-dihydro-5H-pyrrolo[3,4-d]pyrimidine-based PARP1/ATR dual inhibitors

基于6,7-二氢-5H-吡咯并[3,4-d]嘧啶的PARP1/ATR双重抑制剂的设计、合成及抗乳腺癌活性评价

He, Meng-Lan; Wang, Zong-Hao; Yao, Xia; Ye, Lu-Lu; Du, Bo-Qun; Wang, Chen-Chen; Chen, Yong-Hao; Wang, Xiao-Xian; Luo, Hui; Gao, Yuan; Ye, Xiang-Yang

Tetrandrine regulates NAADP-mediated calcium signaling through a LIMP-2-dependent and sphingosine-mediated mechanism.

四氢黄连碱通过 LIMP-2 依赖性和鞘氨醇介导的机制调节 NAADP 介导的钙信号传导

Chan Wing-Cheung, Zhao Qian, Wong Koon Ho, Tang Hok-Him, Mok Daniel Kam-Wah, Pardeshi Lakhansing, Ruan Ye Chun, Yang Yang, Wong Chi-Ming, Wong Clarence T T, Zhao Yong-Juan, Chan Ka Ying, Yin Zengsheng, Leung Howard Ho-Wai, Ma Xiyang, Chau Mary P, Leung Franco King-Chi, Lui Ying-Ying, Au Shannon Wing-Ngor, Sun Kailei, Mok Chin Yu, Wang Fang, Ma Cong, Ho Yu-Hin, Ye Xiang-Yang, Yeung Man Lung, Zhang Yajing, Zhao Yan Xiang, Liu Jiang, Wong Ka-Hing, Chow Larry M C, Li Xiang David, Tse Gary M, Wong Man-Kin, Shen Xiao, Chiu Pauline, Ko Ben C B

Novel ATR/PARP1 Dual Inhibitors Demonstrate Synergistic Antitumor Efficacy in Triple-Negative Breast Cancer Models.

新型 ATR/PARP1 双重抑制剂在三阴性乳腺癌模型中表现出协同抗肿瘤功效

Gao Yuan, Zhou Jiawei, Wang Chen-Chen, Wang Zong-Hao, Mao Nian-Dong, He Meng-Lan, Zhang Peng-Peng, Huang Ping, Ye Guo-Wei, Zhang Yu-Qing, Tang Feng-Hui, Zhang Hang, Xie Tian, Ye Xiang-Yang

Prevention and Potential Treatment Strategies for Respiratory Syncytial Virus

呼吸道合胞病毒的预防和潜在治疗策略

Sun, Bo-Wen; Zhang, Peng-Peng; Wang, Zong-Hao; Yao, Xia; He, Meng-Lan; Bai, Rui-Ting; Che, Hao; Lin, Jing; Xie, Tian; Hui, Zi; Ye, Xiang-Yang; Wang, Li-Wei

Recent progress in discovery of novel AAK1 inhibitors: from pain therapy to potential anti-viral agents

新型AAK1抑制剂发现的最新进展:从疼痛治疗到潜在的抗病毒药物

Yuan, Ying-Hui; Mao, Nian-Dong; Duan, Ji-Long; Zhang, Hang; Garrido, Carmen; Lirussi, Frédéric; Gao, Yuan; Xie, Tian; Ye, Xiang-Yang

Design, synthesis and biological evaluation of novel histone deacetylase (HDAC) inhibitors derived from β-elemene scaffold

基于β-榄香烯骨架的新型组蛋白去乙酰化酶(HDAC)抑制剂的设计、合成和生物学评价

Gao, Yuan; Duan, Jilong; Dang, Xiawen; Yuan, Yinghui; Wang, Yu; He, Xingrui; Bai, Renren; Ye, Xiang-Yang; Xie, Tian

Nickel-catalyzed cross-electrophile allylation of vinyl bromides and the modification of anti-tumour natural medicine β-elemene

镍催化乙烯基溴化物交叉亲电烯丙基化反应及其对天然抗肿瘤药物β-榄香烯的修饰

Ye, Yang; Qi, Xiang; Xu, Bing; Lin, Ying; Xiang, Huan; Zou, Liang; Ye, Xiang-Yang; Xie, Tian

Races of small molecule clinical trials for the treatment of COVID-19: An up-to-date comprehensive review

治疗 COVID-19 的小分子临床试验竞赛:最新综合综述

Hu, Suwen; Jiang, Songwei; Qi, Xiang; Bai, Renren; Ye, Xiang-Yang; Xie, Tian

Nickel-catalyzed enantioselective 1,2-vinylboration of styrenes

镍催化苯乙烯的对映选择性1,2-乙烯基硼化反应

Ye, Yang; Liu, Jiandong; Xu, Bing; Jiang, Songwei; Bai, Renren; Li, Shijun; Xie, Tian; Ye, Xiang-Yang

Anti-Tumor Drug Discovery Based on Natural Product β-Elemene: Anti-Tumor Mechanisms and Structural Modification

基于天然产物β-榄香烯的抗肿瘤药物发现:抗肿瘤机制和结构修饰

Bai, Ziqiang; Yao, Chuansheng; Zhu, Junlong; Xie, Yuanyuan; Ye, Xiang-Yang; Bai, Renren; Xie, Tian