日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

TNG908 is a brain-penetrant, MTA-cooperative PRMT5 inhibitor developed for the treatment of MTAP-deleted cancers

TNG908 是一种可穿透血脑屏障的 MTA 协同 PRMT5 抑制剂,专为治疗 MTAP 缺失型癌症而开发。

Briggs, Kimberly J; Cottrell, Kevin M; Tonini, Matthew R; Tsai, Alice; Zhang, Minjie; Whittington, Douglas A; Zhang, Wenhai; Lombardo, Steven A; Yoda, Satoshi; Wilker, Erik W; Meier, Samuel R; Yu, Yi; Teng, Teng; Huang, Alan; Maxwell, John P

MET Alterations Are a Recurring and Actionable Resistance Mechanism in ALK-Positive Lung Cancer

MET改变是ALK阳性肺癌中一种反复出现且可靶向治疗的耐药机制

Dagogo-Jack, Ibiayi; Yoda, Satoshi; Lennerz, Jochen K; Langenbucher, Adam; Lin, Jessica J; Rooney, Marguerite M; Prutisto-Chang, Kylie; Oh, Audris; Adams, Nathaniel A; Yeap, Beow Y; Chin, Emily; Do, Andrew; Marble, Hetal D; Stevens, Sara E; Digumarthy, Subba R; Saxena, Ashish; Nagy, Rebecca J; Benes, Cyril H; Azzoli, Christopher G; Lawrence, Michael S; Gainor, Justin F; Shaw, Alice T; Hata, Aaron N

Small cell transformation of ROS1 fusion-positive lung cancer resistant to ROS1 inhibition

对 ROS1 抑制剂耐药的 ROS1 融合阳性肺癌的小细胞转化

Lin, Jessica J; Langenbucher, Adam; Gupta, Pranav; Yoda, Satoshi; Fetter, Isobel J; Rooney, Marguerite; Do, Andrew; Kem, Marina; Chang, Kylie Prutisto; Oh, Audris Y; Chin, Emily; Juric, Dejan; Corcoran, Ryan B; Dagogo-Jack, Ibiayi; Gainor, Justin F; Stone, James R; Lennerz, Jochen K; Lawrence, Michael S; Hata, Aaron N; Mino-Kenudson, Mari; Shaw, Alice T

Landscape of Acquired Resistance to Osimertinib in EGFR-Mutant NSCLC and Clinical Validation of Combined EGFR and RET Inhibition with Osimertinib and BLU-667 for Acquired RET Fusion

EGFR突变型非小细胞肺癌中奥希替尼获得性耐药的现状及奥希替尼联合BLU-667治疗获得性RET融合的EGFR和RET联合抑制的临床验证

Piotrowska, Zofia; Isozaki, Hideko; Lennerz, Jochen K; Gainor, Justin F; Lennes, Inga T; Zhu, Viola W; Marcoux, Nicolas; Banwait, Mandeep K; Digumarthy, Subba R; Su, Wenjia; Yoda, Satoshi; Riley, Amanda K; Nangia, Varuna; Lin, Jessica J; Nagy, Rebecca J; Lanman, Richard B; Dias-Santagata, Dora; Mino-Kenudson, Mari; Iafrate, A John; Heist, Rebecca S; Shaw, Alice T; Evans, Erica K; Clifford, Corinne; Ou, Sai-Hong I; Wolf, Beni; Hata, Aaron N; Sequist, Lecia V

Patterns of Metastatic Spread and Mechanisms of Resistance to Crizotinib in ROS1-Positive Non-Small-Cell Lung Cancer

ROS1阳性非小细胞肺癌的转移扩散模式及对克唑替尼的耐药机制

Gainor, Justin F; Tseng, Diane; Yoda, Satoshi; Dagogo-Jack, Ibiayi; Friboulet, Luc; Lin, Jessica J; Hubbeling, Harper G; Dardaei, Leila; Farago, Anna F; Schultz, Katherine R; Ferris, Lorin A; Piotrowska, Zofia; Hardwick, James; Huang, Donghui; Mino-Kenudson, Mari; Iafrate, A John; Hata, Aaron N; Yeap, Beow Y; Shaw, Alice T

Molecular Mechanisms of Resistance to First- and Second-Generation ALK Inhibitors in ALK-Rearranged Lung Cancer.

ALK重排肺癌对第一代和第二代ALK抑制剂产生耐药性的分子机制

Gainor Justin F, Dardaei Leila, Yoda Satoshi, Friboulet Luc, Leshchiner Ignaty, Katayama Ryohei, Dagogo-Jack Ibiayi, Gadgeel Shirish, Schultz Katherine, Singh Manrose, Chin Emily, Parks Melissa, Lee Dana, DiCecca Richard H, Lockerman Elizabeth, Huynh Tiffany, Logan Jennifer, Ritterhouse Lauren L, Le Long P, Muniappan Ashok, Digumarthy Subba, Channick Colleen, Keyes Colleen, Getz Gad, Dias-Santagata Dora, Heist Rebecca S, Lennerz Jochen, Sequist Lecia V, Benes Cyril H, Iafrate A John, Mino-Kenudson Mari, Engelman Jeffrey A, Shaw Alice T

Deregulation of histone lysine methyltransferases contributes to oncogenic transformation of human bronchoepithelial cells

组蛋白赖氨酸甲基转移酶的失调促进人支气管上皮细胞的癌变转化

Watanabe, Hideo; Soejima, Kenzo; Yasuda, Hiroyuki; Kawada, Ichiro; Nakachi, Ichiro; Yoda, Satoshi; Naoki, Katsuhiko; Ishizaka, Akitoshi