日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-Guided Optimization of 4-Chloro-Pyrazolopyridine Analogs for Covalent PREP Inhibition

基于结构的4-氯吡唑并吡啶类似物优化用于共价PREP抑制

Thakur, Kalyani; Fucci, Ian; Pandian, Joshua; Suazo, Kiall F; Monteiro, Diana C F; Yoo, Euna

Granzyme B-Targeting Quenched Activity-Based Probes for Assessing Tumor Response to Immunotherapy

靶向颗粒酶B的淬灭活性探针用于评估肿瘤对免疫疗法的反应

Kazim, Muhammad; Ganguly, Arghya; Malespini, Sebastian M; Thang, Lai; Patel, Nimit L; Kim, Caleb; Thakur, Kalyani; Kalen, Joseph D; Calcagno, Claudia; Difilippantonio, Simone; Yoo, Euna

A robust fluorogenic substrate for chikungunya virus protease (nsP2) activity

一种用于检测基孔肯雅病毒蛋白酶(nsP2)活性的强效荧光底物

Makhaik, Sparsh; Rut, Wioletta; Choudhary, Shruti; Upadhyay, Tulsi; Hao, Chenzhou; Westberg, Michael; Bobst, Cedric; Yoo, Euna; Fejzo, Jasna; Lin, Michael Z; Bogyo, Matthew; Thompson, Paul; Drag, Marcin; Hardy, Jeanne A

Development of Granzyme A Turn-ON Fluorescent Activity-Based Probes

基于颗粒酶A开启荧光活性的探针的开发

Malespini, Sebastian M; Kazim, Muhammad; Yoo, Euna

A Robust Fluorogenic Substrate for Chikungunya Virus Protease (nsP2) Activity

一种用于检测基孔肯雅病毒蛋白酶 (nsP2) 活性的强效荧光底物

Makhaik, Sparsh; Rut, Wioletta; Choudhary, Shruti; Upadhyay, Tulsi; Hao, Chenzhou; Westberg, Michael; Bobst, Cedric; Yoo, Euna; Fejzo, Jasna; Lin, Michael Z; Bogyo, Matthew; Thompson, Paul; Drag, Marcin; Hardy, Jeanne A

Granzyme-targeting quenched activity-based probes for assessing tumor response to immunotherapy

靶向颗粒酶的淬灭活性探针用于评估肿瘤对免疫疗法的反应

Kazim, Muhammad; Ganguly, Arghya; Malespini, Sebastian M; Thang, Lai; Patel, Nimit L; Kim, Caleb; Kalen, Joseph D; Difilippantonio, Simone; Yoo, Euna

Discovery of a Tunable Heterocyclic Electrophile 4-Chloro-pyrazolopyridine That Defines a Unique Subset of Ligandable Cysteines

发现一种可调控的杂环亲电试剂 4-氯吡唑并吡啶,它定义了可配位半胱氨酸的一个独特子集

Kim, Hong-Rae; Byun, David P; Thakur, Kalyani; Ritchie, Jennifer; Xie, Yixin; Holewinski, Ronald; Suazo, Kiall F; Stevens, Mckayla; Liechty, Hope; Tagirasa, Ravichandra; Jing, Yihang; Andresson, Thorkell; Johnson, Steven M; Yoo, Euna

Covalent Inhibition by a Natural Product-Inspired Latent Electrophile

天然产物启发式潜在亲电试剂的共价抑制

Byun, David P; Ritchie, Jennifer; Jung, Yejin; Holewinski, Ronald; Kim, Hong-Rae; Tagirasa, Ravichandra; Ivanic, Joseph; Weekley, Claire M; Parker, Michael W; Andresson, Thorkell; Yoo, Euna

Self-assembled adipose-derived mesenchymal stem cells as an extracellular matrix component- and growth factor-enriched filler

自组装脂肪间充质干细胞作为细胞外基质成分和生长因子富集的填充剂

Choa Park, Ok-Hee Lee, Jin Ju Park, Jiyoon Yoo, Euna Kwon, Jie-Eun Park, Byeong-Cheol Kang, Dong-Sup Lee, Jaejin Cho

Covalent Macrocyclic Proteasome Inhibitors Mitigate Resistance in Plasmodium falciparum

共价大环蛋白酶体抑制剂可减轻恶性疟原虫的耐药性

Bennett, John M; Ward, Kurt E; Muir, Ryan K; Kabeche, Stephanie; Yoo, Euna; Yeo, Tomas; Lam, Grace; Zhang, Hao; Almaliti, Jehad; Berger, Gabriel; Faucher, Franco F; Lin, Gang; Gerwick, William H; Yeh, Ellen; Fidock, David A; Bogyo, Matthew