日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Benzoxazole Derivatives as Potent FXR and PPARα Dual Agonists With Anti-Fibrotic and Metabolic Regulatory Effects

苯并恶唑衍生物作为强效FXR和PPARα双重激动剂,具有抗纤维化和代谢调节作用

Kim, Mi-Jeong; Han, Dong-Gyun; Park, Hyeon Seo; Ha, Sugyeong; Noh, Sang Gyun; Kim, Jeongwon; Yoo, Ji-An; Kim, Byeong Moo; Battogtokh, Khas-Erdene; Oh, Soohwan; Jung, Youngmi; Jung, Youngsuk; Chung, Hae Young; Moon, Hyung Ryong; Yoon, In-Soo; Chung, Ki Wung

Carbutamide, an Obsolete Anti-Diabetic Drug, Has Potential as a Potent Anticolitic Agent via Azo-Conjugation with Mesalazine

卡巴汀是一种已停用的抗糖尿病药物,可通过与美沙拉嗪偶联,成为一种强效抗结肠炎药物。

Ju, Sanghyun; Kim, Suji; Kim, Taeyoung; Yoo, Jin-Wook; Yoon, In-Soo; Kim, Eunsoo; Jung, Yunjin

Pharmacokinetic and Bioequivalence Evaluation of Two Sitagliptin Tablets With Different Salts in Healthy Subjects

在健康受试者中对两种不同盐类的西格列汀片剂进行药代动力学和生物等效性评价

Hyun, Usok; Chu, Seongnam; Kim, Sungyun; Hong, Jung-Ki; Kim, Taeyoung; Yoon, In-Soo; Kim, Jung-Jin; Cho, Hyun-Jong

Factors determining the oral absorption and systemic disposition of zeaxanthin in rats: in vitro, in situ, and in vivo evaluations

影响大鼠口服吸收和全身分布的因素:体外、体内和体内评价

Seo, Seong-Wook; Han, Dong-Gyun; Choi, Eugene; Seo, Min-Jeong; Song, Im-Sook; Yoon, In-Soo

Investigation of the Factors Responsible for the Poor Oral Bioavailability of Acacetin in Rats: Physicochemical and Biopharmaceutical Aspects

对导致大鼠口服阿卡西汀生物利用度低的因素进行研究:理化和生物药剂学方面

Han, Dong-Gyun; Cha, Eunju; Joo, Jeongmin; Hwang, Ji Sun; Kim, Sanghyun; Park, Taeuk; Jeong, Yoo-Seong; Maeng, Han-Joo; Kim, Sang-Bum; Yoon, In-Soo

Assessment of Metabolic Interaction between Repaglinide and Quercetin via Mixed Inhibition in the Liver: In Vitro and In Vivo

通过肝脏混合抑制作用评估瑞格列奈与槲皮素的代谢相互作用:体外和体内研究

Kim, Ji-Min; Seo, Seong-Wook; Han, Dong-Gyun; Yun, Hwayoung; Yoon, In-Soo

A Tumor-Immune Interaction Model for Synergistic Combinations of Anti PD-L1 and Ionizing Irradiation Treatment

抗PD-L1疗法与电离辐射治疗协同作用的肿瘤免疫相互作用模型

Byun, Jong Hyuk; Yoon, In-Soo; Jeong, Yong Dam; Kim, Sungchan; Jung, Il Hyo

Preparation and Evaluation of Amino Acid Conjugates of Celecoxib as Prodrugs to Improve the Pharmacokinetic and Therapeutic Properties of Celecoxib

制备和评价塞来昔布氨基酸缀合物作为前药以改善塞来昔布的药代动力学和治疗特性

Lee, Yonghyun; Kim, Jungyun; Kim, Wooseong; Yoon, In-Soo; Jung, Yunjin

Mitigating Effects of Liriope platyphylla on Nicotine-Induced Behavioral Sensitization and Quality Control of Compounds

白麦冬对尼古丁诱导行为致敏的缓解作用及化合物的质量控制

Dahye Yoon, In Soo Ryu, Woo Cheol Shin, Minhan Ka, Hyoung-Geun Kim, Eun Young Jang, Oc-Hee Kim, Young-Seob Lee, Joung-Wook Seo, Dae Young Lee

Pharmacokinetic Evaluation of Metabolic Drug Interactions between Repaglinide and Celecoxib by a Bioanalytical HPLC Method for Their Simultaneous Determination with Fluorescence Detection

采用生物分析高效液相色谱法结合荧光检测法同时测定瑞格列奈和塞来昔布的代谢药物相互作用,进行药代动力学评价

Han, Dong-Gyun; Kwak, Jinsook; Seo, Seong-Wook; Kim, Ji-Min; Yoo, Jin-Wook; Jung, Yunjin; Lee, Yun-Hee; Kim, Min-Soo; Jung, Young-Suk; Yun, Hwayoung; Yoon, In-Soo