日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

New Adamantane-Containing Edaravone Conjugates as Potential Neuroprotective Agents for ALS Treatments

含有金刚烷的新型依达拉奉结合物可作为 ALS 治疗的潜在神经保护剂

Maria A Lapshina, Elena F Shevtsova, Vladimir V Grigoriev, Aleksey Yu Aksinenko, Aleksey A Ustyugov, Daniil A Steinberg, Grigoriy V Maleev, Elena S Dubrovskaya, Tatiana V Goreva, Tatiana A Epishina, Vladimir L Zamoyski, Galina F Makhaeva, Vladimir P Fisenko, Ivan M Veselov, Daria V Vinogradova, Serg

Conjugates of Methylene Blue with Cycloalkaneindoles as New Multifunctional Agents for Potential Treatment of Neurodegenerative Disease

亚甲蓝与环烷吲哚的结合物作为治疗神经退行性疾病的新型多功能药物

Sergey O Bachurin, Elena F Shevtsova, Galina F Makhaeva, Alexey Yu Aksinenko, Vladimir V Grigoriev, Tatiana V Goreva, Tatiana A Epishina, Nadezhda V Kovaleva, Natalia P Boltneva, Sofya V Lushchekina, Elena V Rudakova, Darya V Vinogradova, Pavel N Shevtsov, Elena A Pushkareva, Ludmila G Dubova, Tatia

A bioisostere of Dimebon/Latrepirdine delays the onset and slows the progression of pathology in FUS transgenic mice

Dimebon/Latrepirdine 的生物等排体可延缓 FUS 转基因小鼠病理的发生并减缓其进展。

Chaprov, Kirill; Rezvykh, Alexander; Funikov, Sergei; Ivanova, Tamara A; Lysikova, Ekaterina A; Deykin, Alexei V; Kukharsky, Michail S; Yu Aksinenko, Alexey; Bachurin, Sergey O; Ninkina, Natalia; Buchman, Vladimir L

Conjugation of Aminoadamantane and γ-Carboline Pharmacophores Gives Rise to Unexpected Properties of Multifunctional Ligands

氨基金刚烷与 γ-咔啉药效团的结合产生意想不到的多功能配体特性

Sergey O Bachurin, Galina F Makhaeva, Elena F Shevtsova, Alexey Yu Aksinenko, Vladimir V Grigoriev, Pavel N Shevtsov, Tatiana V Goreva, Tatiana A Epishina, Nadezhda V Kovaleva, Elena A Pushkareva, Natalia P Boltneva, Sofya V Lushchekina, Alexey V Gabrelyan, Vladimir L Zamoyski, Lyudmila G Dubova, El

Conjugates of methylene blue with γ-carboline derivatives as new multifunctional agents for the treatment of neurodegenerative diseases

亚甲蓝与γ-咔啉衍生物的结合物作为治疗神经退行性疾病的新型多功能药物

Sergey O Bachurin, Galina F Makhaeva, Elena F Shevtsova, Natalia P Boltneva, Nadezhda V Kovaleva, Sofya V Lushchekina, Elena V Rudakova, Ludmila G Dubova, Daria V Vinogradova, Vladimir B Sokolov, Alexey Yu Aksinenko, Vladimir P Fisenko, Rudy J Richardson, Gjumrakch Aliev

Novel conjugates of aminoadamantanes with carbazole derivatives as potential multitarget agents for AD treatment

氨基金刚烷与咔唑衍生物的新型结合物可作为 AD 治疗的潜在多靶点药物

Sergey O Bachurin, Elena F Shevtsova, Galina F Makhaeva, Vladimir V Grigoriev, Natalia P Boltneva, Nadezhda V Kovaleva, Sofya V Lushchekina, Pavel N Shevtsov, Margarita E Neganova, Olga M Redkozubova, Elena V Bovina, Alexey V Gabrelyan, Vladimir P Fisenko, Vladimir B Sokolov, Alexey Yu Aksinenko, Va

Conjugates of γ-Carbolines and Phenothiazine as new selective inhibitors of butyrylcholinesterase and blockers of NMDA receptors for Alzheimer Disease

γ-咔啉与吩噻嗪的结合物作为丁酰胆碱酯酶的新型选择性抑制剂和阿尔茨海默病的 NMDA 受体阻滞剂

Galina F Makhaeva, Sofya V Lushchekina, Natalia P Boltneva, Vladimir B Sokolov, Vladimir V Grigoriev, Olga G Serebryakova, Ekaterina A Vikhareva, Alexey Yu Aksinenko, George E Barreto, Gjumrakch Aliev, Sergey O Bachurin