日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-based design of an opioid receptor modulator for enhanced morphine analgesia

基于结构的阿片受体调节剂设计及其在增强吗啡镇痛中的应用

Wang, Yue; Luo, Ping; Xu, Haiyan; Zhan, Li; Sakamoto, Kensuke; Li, Mingyu; Wang, Jing; Huang, Xi-Ping; Zhou, Jianhui; Liu, Tao; Suo, Yanrui; Fan, Wenjia; He, Xinheng; Xu, Youwei; Cai, Yongjie; Wang, Chao; Zhao, Yuxi; Dai, Antao; Lai, Yali; Yuan, Qingning; Hu, Wen; Wu, Kai; Yang, Dehua; Cheng, Xi; Lu, Xiaojie; Krumm, Brian; Kenakin, Terry; Zhang, Jian; Roth, Bryan L; Gao, Zhaobing; Xu, H Eric; Zhuang, Youwen

Structural insight into GPR55 ligand recognition and G-protein coupling

GPR55配体识别和G蛋白偶联的结构解析

Xia, Ruixue; Yuan, Qingning; Wang, Na; Hou, Li; Abe, Junpei; Song, Jing; Ito, Yukishige; Xu, H Eric; He, Yuanzheng

Molecular mechanism of the arrestin-biased agonism of neurotensin receptor 1 by an intracellular allosteric modulator

细胞内变构调节剂介导的神经降压素受体1的阻遏蛋白偏向性激动作用的分子机制

Sun, Demeng; Li, Xiang; Yuan, Qingning; Wang, Yuanxia; Shi, Pan; Zhang, Huanhuan; Wang, Tao; Sun, Wenjing; Ling, Shenglong; Liu, Yuanchun; Lai, Jinglin; Xie, Wenqin; Yin, Wanchao; Liu, Lei; Xu, H Eric; Tian, Changlin

Structural insights into the agonist activity of the nonpeptide modulator JR14a on C3aR

非肽类调节剂JR14a对C3aR激动剂活性的结构解析

Luo, Ping; Xin, Wenwen; Guo, Shimeng; Li, Xin; Zhang, Qing; Xu, Youwei; He, Xinheng; Wang, Yue; Fan, Wenjia; Yuan, Qingning; Wu, Kai; Hu, Wen; Zhuang, Youwen; Xu, H Eric; Xie, Xin

Molecular mechanisms of urate transport by the native human URAT1 and its inhibition by anti-gout drugs

人体内天然URAT1转运尿酸的分子机制及其被抗痛风药物抑制的机制

Wu, Canrong; Zhang, Chao; Jin, Sanshan; Wang, James Jiqi; Dai, Antao; Xu, Jiuyin; Zhang, Heng; Yang, Xuemei; He, Xinheng; Yuan, Qingning; Hu, Wen; Xu, Youwei; Wang, Mingwei; Jiang, Yi; Yang, Dehua; Xu, H Eric

Molecular basis for ligand recognition and receptor activation of the prostaglandin D2 receptor DP1.

前列腺素D2受体DP1的配体识别和受体激活的分子基础

Xu Jiuyin, Wu Yanli, Xu Youwei, Li Yang, He Xinheng, Zhang Heng, Wang James Jiqi, Hou Jingjing, Li Junrui, Hu Wen, Wu Kai, Yuan Qingning, Wu Canrong, Xu H Eric

Structural insights into hormone recognition and G-protein coupling of the urotensin-II receptor

尿张素II受体激素识别和G蛋白偶联的结构解析

Gao, Tianyu; You, Chongzhao; Cao, Yinglong; Xu, Xiaofang; Yuan, Qingning; Shen, Shiyi; Xu, H Eric; Duan, Jia

Bitter taste receptor TAS2R14 activation and G protein assembly by an intracellular agonist

细胞内激动剂激活苦味受体TAS2R14并组装G蛋白

Tao, Lele; Wang, Dongxue; Yuan, Qingning; Zhao, Fenghui; Zhang, Yu; Du, Tianyuan; Shen, Shiyi; Xu, H Eric; Li, Yi; Yang, Dehua; Duan, Jia

Mechanisms of ligand recognition and activation of melanin-concentrating hormone receptors

黑色素浓缩激素受体的配体识别和激活机制

He, Qian; Yuan, Qingning; Shan, Hong; Wu, Canrong; Gu, Yimin; Wu, Kai; Hu, Wen; Zhang, Yumu; He, Xinheng; Xu, H Eric; Zhao, Li-Hua

Structural insights into the triple agonism at GLP-1R, GIPR and GCGR manifested by retatrutide

瑞他曲肽对 GLP-1R、GIPR 和 GCGR 的三重激动作用的结构解析

Li, Wenzhuo; Zhou, Qingtong; Cong, Zhaotong; Yuan, Qingning; Li, Wenxin; Zhao, Fenghui; Xu, H Eric; Zhao, Li-Hua; Yang, Dehua; Wang, Ming-Wei