Discovery of the Orally Effective Thyrotropin-Releasing Hormone Mimetic: 1-{ N-[(4 S,5 S)-(5-Methyl-2-oxooxazolidine-4-yl)carbonyl]-3-(thiazol-4-yl)-l-alanyl}-(2 R)-2-methylpyrrolidine Trihydrate (Rovatirelin Hydrate)
发现口服有效的促甲状腺激素释放激素模拟物:1-{N-[(4S,5S)-(5-甲基-2-氧代恶唑烷-4-基)羰基]-3-(噻唑-4-基)-l-丙氨酰}-(2R)-2-甲基吡咯烷三水合物(罗伐替林水合物)
期刊:ACS Omega
影响因子:3.7
doi:10.1021/acsomega.8b01481
Naotake Kobayashi, Norihito Sato, Yuko Fujimura, Tsuyoshi Kihara, Katsuji Sugita, Kouji Takahashi, Katsumi Koike, Tamio Sugawara, Yukio Tada, Hiroshi Nakai, Takayoshi Yoshikawa