Mitoxantrone inhibits and downregulates ER α through binding at the DBD-LBD interface
米托蒽醌通过与DNA结合域(DBD)-配体结合域(LBD)界面结合,抑制并下调雌激素受体α(ERα)。
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影响因子:
doi:10.1101/2025.01.07.631371
Wang, Han; Luo, Yuxuan; Artham, Sandeep; Wang, Qianqian; Peng, Yi; Yun, Zixi; Li, Xinyue; Wu, Chen; Liu, Zhenghao; Weber-Bonk, Kristen L; Pai, Chun-Peng; Cao, Yuan; Yue, Jiangan; Park, Sunghee; Keri, Ruth A; Geng, Lisheng; McDonnell, Donald P; Kao, Hung-Ying; Yang, Sichun