日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Dichloroacetate, a pyruvate dehydrogenase kinase inhibitor, ameliorates type 2 diabetes via reduced gluconeogenesis

二氯乙酸是一种丙酮酸脱氢酶激酶抑制剂,可通过减少糖异生来改善 2 型糖尿病

Yuko Katayama, Yayoi Kawata, Yusuke Moritoh, Masanori Watanabe

The enzymatic activity of inositol hexakisphosphate kinase controls circulating phosphate in mammals

肌醇六磷酸激酶的酶活性控制哺乳动物体内循环磷酸盐的水平。

Yusuke Moritoh,Shin-Ichi Abe,Hiroki Akiyama,Akihiro Kobayashi,Ryokichi Koyama,Ryoma Hara,Shizuo Kasai,Masanori Watanabe

SCO-267, a GPR40 Full Agonist, Stimulates Islet and Gut Hormone Secretion and Improves Glycemic Control in Humans

SCO-267 是一种 GPR40 完全激动剂,可刺激胰岛和肠道激素分泌并改善人类血糖控制

Harunobu Nishizaki, Osamu Matsuoka, Tomoya Kagawa, Akihiro Kobayashi, Masanori Watanabe, Yusuke Moritoh

Enteropeptidase inhibition improves kidney function in a rat model of diabetic kidney disease

肠肽酶抑制可改善糖尿病肾病大鼠模型的肾功能

Jun Sugama, Yuko Katayama, Yusuke Moritoh, Masanori Watanabe

SCO-792, an enteropeptidase inhibitor, improves disease status of diabetes and obesity in mice

肠肽酶抑制剂 SCO-792 改善小鼠糖尿病和肥胖症的病情

Hiroaki Yashiro, Kenichi Hamagami, Hideyuki Hiyoshi, Jun Sugama, Kazue Tsuchimori, Fuminari Yamaguchi, Yusuke Moritoh, Minoru Sasaki, Tsuyoshi Maekawa, Yukio Yamada, Masanori Watanabe

Discovery and characterization of a small-molecule enteropeptidase inhibitor, SCO-792

小分子肠肽酶抑制剂 SCO-792 的发现和表征

Masako Sasaki, Ikuo Miyahisa, Sachiko Itono, Hiroaki Yashiro, Hideyuki Hiyoshi, Kazue Tsuchimori, Ken-Ichi Hamagami, Yusuke Moritoh, Masanori Watanabe, Kimio Tohyama, Minoru Sasaki, Jun-Ichi Sakamoto, Tomohiro Kawamoto

GPR40 full agonism exerts feeding suppression and weight loss through afferent vagal nerve

GPR40 完全激动剂通过传入迷走神经发挥摄食抑制和减肥作用

Hikaru Ueno, Ryo Ito, Shin-Ichi Abe, Hitomi Ogino, Minoru Maruyama, Hirohisa Miyashita, Yasufumi Miyamoto, Yusuke Moritoh, Yoshiyuki Tsujihata, Koji Takeuchi, Nobuhiro Nishigaki

GLP-1 suppresses glucagon secretion in human pancreatic alpha-cells by inhibition of P/Q-type Ca2+ channels

GLP-1 通过抑制 P/Q 型 Ca2+ 通道来抑制人类胰腺 α 细胞中的胰高血糖素分泌

Reshma Ramracheya, Caroline Chapman, Margarita Chibalina, Haiqiang Dou, Caroline Miranda, Alejandro González, Yusuke Moritoh, Makoto Shigeto, Quan Zhang, Matthias Braun, Anne Clark, Paul R Johnson, Patrik Rorsman, Linford J B Briant

Inositol Hexakisphosphate Kinase 3 Regulates Metabolism and Lifespan in Mice

肌醇六磷酸激酶3调节小鼠的代谢和寿命

Yusuke Moritoh,Masahiro Oka,Yoshitaka Yasuhara,Hiroyuki Hozumi,Kimihiko Iwachidow,Hiromitsu Fuse,Ryuichi Tozawa

GLP-1 inhibits and adrenaline stimulates glucagon release by differential modulation of N- and L-type Ca2+ channel-dependent exocytosis

GLP-1 通过对 N 型和 L 型 Ca2+ 通道依赖性胞吐的差异调节来抑制胰高血糖素释放,而肾上腺素则刺激胰高血糖素释放

Yang Z De Marinis #, Albert Salehi #, Caroline E Ward #, Quan Zhang #, Fernando Abdulkader, Martin Bengtsson, Orit Braha, Matthias Braun, Reshma Ramracheya, Stefan Amisten, Abdella M Habib, Yusuke Moritoh, Enming Zhang, Frank Reimann, Anders Rosengren, Tadao Shibasaki, Fiona Gribble, Erik Renström,