日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-guided design of partial agonists at an opioid receptor.

基于结构的阿片受体部分激动剂设计

Varga Balazs R, Bernhard Sarah M, El Daibani Amal, Zaidi Saheem A, Lam Jordy H, Aguilar Jhoan, Appourchaux Kevin, Nazarova Antonina L, Kouvelis Alexa, Shinouchi Ryosuke, Hammond Haylee R, Eans Shainnel O, Weinreb Violetta, Margolis Elyssa B, Fay Jonathan F, Huang Xi-Ping, Pradhan Amynah, Katritch Vsevolod, McLaughlin Jay P, Majumdar Susruta, Che Tao

Synthesis and Pharmacology of a Morphinan-Derived Dual Mu-Kappa Opioid Receptor Agonist Analgesic.

吗啡烷衍生的双重μ-κ阿片受体激动剂镇痛药的合成与药理学研究

Varga Balazs R, Uprety Rajendra, Paul Barnali, Knoll Alexis, Ramos-Gonzalez Nokomis, Appourchaux Kevin, Taylor Tori, Turgutalp Bengisu, Shinouchi Ryosuke, Eans Shainnel O, Williams Ashai K, Vasquez-Grinnell Steven G, Zaidi Saheem, Nazarova Antonina L, Varadi Andras, Le Rouzic Valerie, Brown Taylor G, Martinez Shani, Ansonoff Michael, Dardashti Rebecca Notis, Hunkele Amanda, Subrath Joan, Welch Matthew, Xu Jin, Rossi Grace C, Pintar John, Pasternak Gavril W, Katritch Vsevolod, McLaughlin Jay P, Pan Ying Xian, Majumdar Susruta

Structure-guided design of a peripherally restricted chemogenetic system.

结构导向的外周限制性化学遗传系统设计

Kang Hye Jin, Krumm Brian E, Tassou Adrien, Geron Matan, DiBerto Jeffrey F, Kapolka Nicholas J, Gumpper Ryan H, Sakamoto Kensuke, Dewran Kocak D, Olsen Reid H J, Huang Xi-Ping, Zhang Shicheng, Huang Karen L, Zaidi Saheem A, Nguyen MyV T, Jo Min Jeong, Katritch Vsevolod, Fay Jonathan F, Scherrer Grégory, Roth Bryan L

Virtual Screening of a Chemically Diverse "Superscaffold" Library Enables Ligand Discovery for a Key GPCR Target

利用化学结构多样的“超级骨架”库进行虚拟筛选,可发现关键GPCR靶点的配体

Grotsch, Katharina; Sadybekov, Anastasiia V; Hiller, Sydney; Zaidi, Saheem; Eremin, Dmitry; Le, Austen; Liu, Yongfeng; Smith, Evan Carlton; Illiopoulis-Tsoutsouvas, Christos; Thomas, Joice; Aggarwal, Shubhangi; Pickett, Julie E; Reyes, Cesar; Picazo, Elias; Roth, Bryan L; Makriyannis, Alexandros; Katritch, Vsevolod; Fokin, Valery V

Structure-based design of bitopic ligands for the µ-opioid receptor

基于结构的μ-阿片受体双位点配体设计

Faouzi, Abdelfattah; Wang, Haoqing; Zaidi, Saheem A; DiBerto, Jeffrey F; Che, Tao; Qu, Qianhui; Robertson, Michael J; Madasu, Manish K; El Daibani, Amal; Varga, Balazs R; Zhang, Tiffany; Ruiz, Claudia; Liu, Shan; Xu, Jin; Appourchaux, Kevin; Slocum, Samuel T; Eans, Shainnel O; Cameron, Michael D; Al-Hasani, Ream; Pan, Ying Xian; Roth, Bryan L; McLaughlin, Jay P; Skiniotis, Georgios; Katritch, Vsevolod; Kobilka, Brian K; Majumdar, Susruta

Harnessing Ion-Binding Sites for GPCR Pharmacology

利用离子结合位点进行GPCR药理学研究

Zarzycka, Barbara; Zaidi, Saheem A; Roth, Bryan L; Katritch, Vsevolod

Dynamic Strategic Bond Analysis Yields a Ten-Step Synthesis of 20-nor-Salvinorin A, a Potent κ-OR Agonist

动态战略键分析得出强效κ-阿片受体激动剂20-去甲-萨尔维诺林A的十步合成路线

Roach, Jeremy J; Sasano, Yusuke; Schmid, Cullen L; Zaidi, Saheem; Katritch, Vsevolod; Stevens, Raymond C; Bohn, Laura M; Shenvi, Ryan A

Understanding molecular interactions between scavenger receptor A and its natural product inhibitors through molecular modeling studies.

通过分子建模研究了解清道夫受体 A 与其天然产物抑制剂之间的分子相互作用

Pagare Piyusha P, Zaidi Saheem A, Zhang Xiaomei, Li Xia, Yu Xiaofei, Wang Xiang-Yang, Zhang Yan

Small molecule inhibits activity of scavenger receptor A: Lead identification and preliminary studies

小分子抑制清道夫受体A的活性:先导化合物筛选和初步研究

Yuan, Yunyun; Li, Xia; Zaidi, Saheem A; Arnatt, Christopher K; Yu, Xiaofei; Guo, Chunqing; Wang, Xiang-Yang; Zhang, Yan

5-Hydroxy-2-(2-phenylethyl)chromone (5-HPEC): a novel non-nitrogenous ligand for 5-HT2B receptor

5-羟基-2-(2-苯乙基)色酮 (5-HPEC):一种新型的5-HT2B受体非含氮配体

Williams, Dwight A; Zaidi, Saheem A; Zhang, Yan