Novel K-Ras G12C Switch-II Covalent Binders Destabilize Ras and Accelerate Nucleotide Exchange
新型 K-Ras G12C Switch-II 共价结合剂可使 Ras 不稳定并加速核苷酸交换
期刊:Journal of Chemical Information and Modeling
影响因子:5.3
doi:10.1021/acs.jcim.7b00399
Nnadi, Chimno I; Jenkins, Meredith L; Gentile, Daniel R; Bateman, Leslie A; Zaidman, Daniel; Balius, Trent E; Nomura, Daniel K; Burke, John E; Shokat, Kevan M; London, Nir