日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification of Potent Reverse Indazole Inhibitors for HPK1

鉴定HPK1的强效反向吲唑抑制剂

Yu, Elsie C; Methot, Joey L; Fradera, Xavier; Lesburg, Charles A; Lacey, Brian M; Siliphaivanh, Phieng; Liu, Ping; Smith, Dustin M; Xu, Zangwei; Piesvaux, Jennifer A; Kawamura, Shuhei; Xu, Haiyan; Miller, J Richard; Bittinger, Mark; Pasternak, Alexander

Discovery of Diaminopyrimidine Carboxamide HPK1 Inhibitors as Preclinical Immunotherapy Tool Compounds

二氨基嘧啶羧酰胺类HPK1抑制剂作为临床前免疫治疗工具化合物的发现

Vara, Brandon A; Levi, Samuel M; Achab, Abdelghani; Candito, David A; Fradera, Xavier; Lesburg, Charles A; Kawamura, Shuhei; Lacey, Brian M; Lim, Jongwon; Methot, Joey L; Xu, Zangwei; Xu, Haiyan; Smith, Dustin M; Piesvaux, Jennifer A; Miller, J Richard; Bittinger, Mark; Ranganath, Sheila H; Bennett, David J; DiMauro, Erin F; Pasternak, Alexander

Allosteric Modulation of Protein Arginine Methyltransferase 5 (PRMT5)

蛋白质精氨酸甲基转移酶 5 (PRMT5) 的变构调节

Palte, Rachel L; Schneider, Sebastian E; Altman, Michael D; Hayes, Robert P; Kawamura, Shuhei; Lacey, Brian M; Mansueto, My Sam; Reutershan, Michael; Siliphaivanh, Phieng; Sondey, Christopher; Xu, Haiyan; Xu, Zangwei; Ye, Yingchun; Machacek, Michelle R

Pharmacological inhibition of hematopoietic progenitor kinase 1 positively regulates T-cell function

药理学抑制造血祖细胞激酶1可正向调节T细胞功能

Yun Wang ,Kelvin Zhang ,Peter Georgiev ,Steven Wells ,Haiyan Xu ,Brian M Lacey ,Zangwei Xu ,Jason Laskey ,Robbie Mcleod ,Joey L Methot ,Mark Bittinger ,Alexander Pasternak ,Sheila Ranganath

Identification of direct target engagement biomarkers for kinase-targeted therapeutics

鉴定激酶靶向治疗的直接靶点结合生物标志物

Paweletz, Cloud P; Andersen, Jannik N; Pollock, Roy; Nagashima, Kumiko; Hayashi, Mansuo L; Yu, Shangshuan U; Guo, Hongbo; Bobkova, Ekaterina V; Xu, Zangwei; Northrup, Alan; Blume-Jensen, Peter; Hendrickson, Ronald C; Chi, An