日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

In vitro cultured malaria hypnozoites leave a footprint of specific metabolites

体外培养的疟原虫休眠子会留下特定代谢物的痕迹。

Pasini, Erica M; Hakimi, Hassan; Chaiyawong, Nattawat; Klop, Onny; Zeeman, Anne-Marie; Nieuwenhuis, Ivonne; van der Werff, Nicole; Kihara, Kumiko; Kami, Kenjiro; Kocken, Clemens H M; Kaneko, Osamu

Identification of novel compounds with prophylactic activity against hypnozoites using a Plasmodium cynomolgi in vitro model

利用猴疟原虫体外模型鉴定具有预防休眠子活性的新型化合物

Zeeman, Anne-Marie; Vermaat, Lars; Castellote Alvaro, M Isabel; Van der Werff, Nicole M; Glas-Nieuwenhuis, Ivonne G; Harupa-Chung, Anke; Calderón, Félix; Gamo, Fransisco-Javier; Fernandez Alvaro, Elena; Kocken, Clemens H M

Transfection Models to Investigate Plasmodium vivax-Type Dormant Liver Stage Parasites

用于研究间日疟原虫休眠肝期寄生虫的转染模型

Voorberg-van der Wel, Annemarie; Zeeman, Anne-Marie; Kocken, Clemens H M

Metabolic, Pharmacokinetic, and Activity Profile of the Liver Stage Antimalarial (RC-12)

肝期抗疟药(RC-12)的代谢、药代动力学和活性特征

Dong, Yuxiang; Sonawane, Yogesh; Maher, Steven P; Zeeman, Anne-Marie; Chaumeau, Victor; Vantaux, Amélie; Cooper, Caitlin A; Chiu, Francis C K; Ryan, Eileen; McLaren, Jenna; Chen, Gong; Wittlin, Sergio; Witkowski, Benoît; Nosten, François; Sriraghavan, Kamaraj; Kyle, Dennis E; Kocken, Clemens H M; Charman, Susan A; Vennerstrom, Jonathan L

Transcriptional profiling of hepatocytes infected with the replicative form of the malaria parasite Plasmodium cynomolgi

对感染疟原虫复制型(Plasmodium cynomolgi)的肝细胞进行转录组分析

Mitchell, Gabriel; Roma, Guglielmo; Voorberg-van der Wel, Annemarie; Beibel, Martin; Zeeman, Anne-Marie; Schuierer, Sven; Torres, Laura; Flannery, Erika L; Kocken, Clemens H M; Mikolajczak, Sebastian A; Diagana, Thierry T

The Novel bis-1,2,4-Triazine MIPS-0004373 Demonstrates Rapid and Potent Activity against All Blood Stages of the Malaria Parasite

新型双-1,2,4-三嗪化合物MIPS-0004373对疟原虫所有血液阶段均表现出快速而强效的活性

Ellis, Katherine M; Lucantoni, Leonardo; Chavchich, Marina; Abraham, Matthew; De Paoli, Amanda; Luth, Madeline R; Zeeman, Anne-Marie; Delves, Michael J; Terán, Fernando Sánchez-Román; Straschil, Ursula; Baum, Jake; Kocken, Clemens H M; Ralph, Stuart A; Winzeler, Elizabeth A; Avery, Vicky M; Edstein, Michael D; Baell, Jonathan B; Creek, Darren J

Modeling Relapsing Malaria: Emerging Technologies to Study Parasite-Host Interactions in the Liver

复发性疟疾建模:研究肝脏中寄生虫-宿主相互作用的新兴技术

Voorberg-van der Wel, Annemarie; Kocken, Clemens H M; Zeeman, Anne-Marie

Transcriptomic analysis reveals reduced transcriptional activity in the malaria parasite Plasmodium cynomolgi during progression into dormancy

转录组分析揭示,疟原虫(Plasmodium cynomolgi)在进入休眠期过程中转录活性降低。

Bertschi, Nicole L; Voorberg-van der Wel, Annemarie; Zeeman, Anne-Marie; Schuierer, Sven; Nigsch, Florian; Carbone, Walter; Knehr, Judith; Gupta, Devendra K; Hofman, Sam O; van der Werff, Nicole; Nieuwenhuis, Ivonne; Klooster, Els; Faber, Bart W; Flannery, Erika L; Mikolajczak, Sebastian A; Chuenchob, Vorada; Shrestha, Binesh; Beibel, Martin; Bouwmeester, Tewis; Kangwanrangsan, Niwat; Sattabongkot, Jetsumon; Diagana, Thierry T; Kocken, Clemens Hm; Roma, Guglielmo

A tetraoxane-based antimalarial drug candidate that overcomes PfK13-C580Y dependent artemisinin resistance

一种基于四氧烷基的抗疟疾候选药物,可克服 PfK13-C580Y 依赖的青蒿素耐药性。

O'Neill, Paul M; Amewu, Richard K; Charman, Susan A; Sabbani, Sunil; Gnädig, Nina F; Straimer, Judith; Fidock, David A; Shore, Emma R; Roberts, Natalie L; Wong, Michael H-L; Hong, W David; Pidathala, Chandrakala; Riley, Chris; Murphy, Ben; Aljayyoussi, Ghaith; Gamo, Francisco Javier; Sanz, Laura; Rodrigues, Janneth; Cortes, Carolina Gonzalez; Herreros, Esperanza; Angulo-Barturén, Iñigo; Jiménez-Díaz, María Belén; Bazaga, Santiago Ferrer; Martínez-Martínez, María Santos; Campo, Brice; Sharma, Raman; Ryan, Eileen; Shackleford, David M; Campbell, Simon; Smith, Dennis A; Wirjanata, Grennady; Noviyanti, Rintis; Price, Ric N; Marfurt, Jutta; Palmer, Michael J; Copple, Ian M; Mercer, Amy E; Ruecker, Andrea; Delves, Michael J; Sinden, Robert E; Siegl, Peter; Davies, Jill; Rochford, Rosemary; Kocken, Clemens H M; Zeeman, Anne-Marie; Nixon, Gemma L; Biagini, Giancarlo A; Ward, Stephen A

Diversity-oriented synthesis yields novel multistage antimalarial inhibitors.

多样性导向合成产生新型多阶段抗疟疾抑制剂

Kato Nobutaka, Comer Eamon, Sakata-Kato Tomoyo, Sharma Arvind, Sharma Manmohan, Maetani Micah, Bastien Jessica, Brancucci Nicolas M, Bittker Joshua A, Corey Victoria, Clarke David, Derbyshire Emily R, Dornan Gillian L, Duffy Sandra, Eckley Sean, Itoe Maurice A, Koolen Karin M J, Lewis Timothy A, Lui Ping S, Lukens Amanda K, Lund Emily, March Sandra, Meibalan Elamaran, Meier Bennett C, McPhail Jacob A, Mitasev Branko, Moss Eli L, Sayes Morgane, Van Gessel Yvonne, Wawer Mathias J, Yoshinaga Takashi, Zeeman Anne-Marie, Avery Vicky M, Bhatia Sangeeta N, Burke John E, Catteruccia Flaminia, Clardy Jon C, Clemons Paul A, Dechering Koen J, Duvall Jeremy R, Foley Michael A, Gusovsky Fabian, Kocken Clemens H M, Marti Matthias, Morningstar Marshall L, Munoz Benito, Neafsey Daniel E, Sharma Amit, Winzeler Elizabeth A, Wirth Dyann F, Scherer Christina A, Schreiber Stuart L