Antitrypanosomal lead discovery: identification of a ligand-efficient inhibitor of Trypanosoma cruzi CYP51 and parasite growth
抗锥虫药物的先导发现:鉴定出一种克氏锥虫 CYP51 和寄生虫生长的配体有效抑制剂
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/jm400012e
Grasiella Andriani, Emanuele Amata, Joel Beatty, Zeke Clements, Brian J Coffey, Gilles Courtemanche, William Devine, Jessey Erath, Cristin E Juda, Zdzislaw Wawrzak, Jodianne T Wood, Galina I Lepesheva, Ana Rodriguez, Michael P Pollastri