日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

PBRM1 directs PBAF to pericentromeres and protects centromere integrity.

PBRM1 将 PBAF 引导至着丝粒周围区域,从而保护着丝粒的完整性

Lane Karen A, Harrod Alison, Wu Lillian, Roumeliotis Theodoros I, Feng Hugang, Foo Shane, Begg Katheryn A G, Schiavoni Federica, Amin Noa, Zenke Frank T, Melcher Alan A, Choudhary Jyoti S, Downs Jessica A

Semi-mechanistic efficacy model for PARP + ATR inhibitors-application to rucaparib and talazoparib in combination with gartisertib in breast cancer PDXs

PARP + ATR 抑制剂的半机制疗效模型——应用于 rucaparib 和 talazoparib 与 gartisertib 联合治疗乳腺癌 PDX 模型

Villette, Claire C; Dupuy, Nathalie; Brightman, Frances A; Zimmermann, Astrid; Lignet, Floriane; Zenke, Frank T; Terranova, Nadia; Bolleddula, Jayaprakasam; El Bawab, Samer; Chassagnole, Christophe

Author Correction: ATR inhibition augments the efficacy of lurbinectedin in small-cell lung cancer

作者更正:ATR抑制剂可增强鲁比替定在小细胞肺癌中的疗效

Schultz, Christopher W; Zhang, Yang; Elmeskini, Rajaa; Zimmermann, Astrid; Fu, Haiqing; Murai, Yasuhisa; Wangsa, Darawalee; Kumar, Suresh; Takahashi, Nobuyuki; Atkinson, Devon; Saha, Liton Kumar; Lee, Chien-Fei; Elenbaas, Brian; Desai, Parth; Sebastian, Robin; Sharma, Ajit Kumar; Abel, Melissa; Schroeder, Brett; Krishnamurthy, Manan; Bassel, Laurel L; Kumar, Rajesh; Roper, Nitin; Aladjem, Mirit; Zenke, Frank T; Ohler, Zoe Weaver; Pommier, Yves; Thomas, Anish

Mapping combinatorial drug effects to DNA damage response kinase inhibitors

将组合药物效应映射到DNA损伤反应激酶抑制剂

Zhang, Hanrui; Kreis, Julian; Schelhorn, Sven-Eric; Dahmen, Heike; Grombacher, Thomas; Zühlsdorf, Michael; Zenke, Frank T; Guan, Yuanfang

Hyper-Dependence on NHEJ Enables Synergy between DNA-PK Inhibitors and Low-Dose Doxorubicin in Leiomyosarcoma.

对 NHEJ 的过度依赖使得 DNA-PK 抑制剂与低剂量阿霉素在平滑肌肉瘤中产生协同作用

Marino-Enriquez Adrian, Novotny Jan Philipp, Gulhan Doga C, Klooster Isabella, Tran Antuan V, Kasbo Macy, Lundberg Meijun Z, Ou Wen-Bin, Tao Derrick L, Pilco-Janeta Daniel F, Mao Victor Y, Zenke Frank T, Leeper Brittaney A, Gokhale Prafulla C, Cowley Glenn S, Baker Laurence H, Ballman Karla V, Root David E, Albers Joachim, Park Peter J, George Suzanne, Fletcher Jonathan A

ATR represents a therapeutic vulnerability in clear cell renal cell carcinoma

ATR代表了透明细胞肾细胞癌的治疗弱点

Seidel, Philipp; Rubarth, Anne; Zodel, Kyra; Peighambari, Asin; Neumann, Felix; Federkiel, Yannick; Huang, Hsin; Hoefflin, Rouven; Adlesic, Mojca; Witt, Christian; Hoffmann, David J; Metzger, Patrick; Lindemann, Ralph K; Zenke, Frank T; Schell, Christoph; Boerries, Melanie; von Elverfeldt, Dominik; Reichardt, Wilfried; Follo, Marie; Albers, Joachim; Frew, Ian J

Modeling the Effect of Hypoxia and DNA Repair Inhibition on Cell Survival After Photon Irradiation

模拟缺氧和DNA修复抑制对光子照射后细胞存活的影响

Liew, Hans; Klein, Carmen; Zenke, Frank T; Abdollahi, Amir; Debus, Jürgen; Dokic, Ivana; Mairani, Andrea