日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Targeting ERAP1 to disarm Gli activation in Sonic Hedgehog medulloblastoma

靶向ERAP1以抑制Sonic Hedgehog髓母细胞瘤中的Gli激活

Shi, Guoyongyan; Zeqiraj, Elton; Riobo-Del Galdo, Natalia A

High-throughput discovery and characterisation of pentafluorobenzene sulfonamide modifiers of Aurora A kinase

利用高通量方法发现和表征Aurora A激酶的五氟苯磺酰胺修饰剂

Chesti, Julian; Miles, Jennifer A; Collins, Lawrence J; McCallum, Hamish A; Foglizzo, Martina; Ahangar, Mohd Syed; Zeqiraj, Elton; Bayliss, Richard; Warriner, Stuart L; Wright, Megan H; Nelson, Adam

Mechanism and cellular actions of the potent AMPK inhibitor BAY-3827.

强效 AMPK 抑制剂 BAY-3827 的作用机制和细胞作用

Fraguas Bringas Conchita, Ahangar Mohd Syed, Cuenco Joyceline, Liu Hongling, Addinsall Alex B, Lindahl Maria, Ovens Ashley J, Febbraio Mark A, Foretz Marc, Göransson Olga, Scott John W, Zeqiraj Elton, Sakamoto Kei

Systemic Sclerosis Dermal Fibroblast Exosomes Trigger Type 1 Interferon Responses in Keratinocytes via a TBK/JAK/STAT Signaling Axis

系统性硬化症真皮成纤维细胞外泌体通过TBK/JAK/STAT信号轴触发角质形成细胞中的I型干扰素反应

Bryon, Jessica; Wasson, Christopher W; Koeppen, Katja; Chandler, Francesca; Willis, Leon F; Di Donato, Stefano; Klein, Elliott; Zeqiraj, Elton; Ross, Rebecca L; Del Galdo, Francesco

Molecular glues that inhibit deubiquitylase activity and inflammatory signaling.

抑制去泛素化酶活性和炎症信号的分子胶

Chandler Francesca, Reddy Poli Adi Narayana, Bhutda Smita, Ross Rebecca L, Datta Arindam, Walden Miriam, Walker Kieran, Di Donato Stefano, Cassel Joel A, Prakesch Michael A, Aman Ahmed, Datti Alessandro, Campbell Lisa J, Foglizzo Martina, Bell Lillie, Stein Daniel N, Ault James R, Al-Awar Rima S, Calabrese Antonio N, Sicheri Frank, Del Galdo Francesco, Salvino Joseph M, Greenberg Roger A, Zeqiraj Elton

Sequence rules for a long SPOP-binding degron required for protein ubiquitylation

蛋白质泛素化所需的长SPOP结合降解子的序列规则

Makhlouf, Linda; Mishra, Mukul; Makhlouf, Hannah; Manfield, Iain; Busino, Luca; Zeqiraj, Elton

Structure and function of MDM2 and MDM4 in health and disease

MDM2和MDM4在健康和疾病中的结构和功能

Zhu, Ivy Yiyi; Lloyd, Alec; Critchley, William R; Saikia, Queen; Jade, Dhananjay; Divan, Aysha; Zeqiraj, Elton; Harrison, Michael A; Brown, Christopher J; Ponnambalam, Sreenivasan

BRCA1-BARD1 combines multiple chromatin recognition modules to bridge nascent nucleosomes

BRCA1-BARD1 结合多个染色质识别模块,连接新生核小体。

Burdett, Hayden; Foglizzo, Martina; Musgrove, Laura J; Kumar, Dhananjay; Clifford, Gillian; Campbell, Lisa J; Heath, George R; Zeqiraj, Elton; Wilson, Marcus D

Higher-Order Assembly of BRCC36-KIAA0157 Is Required for DUB Activity and Biological Function

BRCC36-KIAA0157 的高级组装是 DUB 活性和生物学功能所必需的

Zeqiraj, Elton; Tian, Lei; Piggott, Christopher A; Pillon, Monica C; Duffy, Nicole M; Ceccarelli, Derek F; Keszei, Alexander F A; Lorenzen, Kristina; Kurinov, Igor; Orlicky, Stephen; Gish, Gerald D; Heck, Albert J R; Guarné, Alba; Greenberg, Roger A; Sicheri, Frank

Structure of an SspH1-PKN1 complex reveals the basis for host substrate recognition and mechanism of activation for a bacterial E3 ubiquitin ligase.

SspH1-PKN1复合物的结构揭示了细菌E3泛素连接酶的宿主底物识别基础和激活机制

Keszei Alexander F A, Tang Xiaojing, McCormick Craig, Zeqiraj Elton, Rohde John R, Tyers Mike, Sicheri Frank