日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Development and Characterization of the First Selective Class IIb Histone Deacetylase Degraders.

首个选择性 IIb 类组蛋白去乙酰化酶降解剂的开发和表征

Zhai Shiyang, Honin Irina, Schäker-Hübner Linda, Hanl Maria, Jacobi Lukas, Dressler Finn, Pieńkowska Dominika Ewa, König Philipp, Gerhartz Jan, Voget Rabea, Bendas Gerd, Gütschow Michael, Meissner Felix, Burckhardt Bjoern B, Nowak Radosław P, Steinebach Christian, Hansen Finn K

Targeted Histone Deacetylase Degradation via Chemical Induced Proximity by Direct Recruitment of the CUL4 Complex Adaptor Protein DDB1

通过化学诱导的邻近效应,直接募集 CUL4 复合物衔接蛋白 DDB1 靶向降解组蛋白去乙酰化酶

Zhai, Shiyang; Willemsen, Nicola; Sun, Tao; Malenica, Mateo; Deng, Shixin; Geyer, Matthias; Hansen, Finn K

Targeted Degradation of Histone Deacetylases via Bypassing E3 Ligase Targeting Chimeras (BYETACs)

通过绕过 E3 连接酶靶向嵌合体 (BYETACs) 靶向降解组蛋白去乙酰化酶

Sun, Tao; Zhai, Shiyang; König, Beate; Honin, Irina; Kponomaizoun, Cindy-Esther; Hansen, Finn K

Light-activatable photochemically targeting chimeras (PHOTACs) enable the optical control of targeted protein degradation of HDAC6

光激活光化学靶向嵌合体(PHOTACs)能够实现对HDAC6靶向蛋白降解的光学控制。

Wurnig, Silas L; Hanl, Maria; Geiger, Thomas M; Zhai, Shiyang; Dressel, Ina; Pieńkowska, Dominika E; Nowak, Radosław P; Hansen, Finn K

DCAF16-Based Covalent Molecular Glues for Targeted Protein Degradation of Histone Deacetylases.

基于DCAF16的共价分子胶用于靶向降解组蛋白去乙酰化酶

Sun Tao, Zhai Shiyang, Lepper Stephan, König Beate, Malenica Mateo, Honin Irina, Hansen Finn K