日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Development of a bioavailable boron-containing PI-103 Bioisostere, PI-103BE

开发一种具有生物利用度的含硼PI-103生物等排体PI-103BE

Luo, Lan; Zhong, Qiu; Guo, Shanchun; Zhang, Changde; Zhang, Qiang; Zheng, Shilong; He, Ling; Wang, Guangdi

Metabolism and Pharmacokinetic Study of the Boron-Containing Prodrug of Belinostat (ZL277), a Pan HDAC Inhibitor with Enhanced Bioavailability.

具有增强生物利用度的泛 HDAC 抑制剂 Belinostat (ZL277) 的含硼前药的代谢和药代动力学研究

Zhang Changde, Guo Shanchun, Zhong Qiu, Zhang Qiang, Hossain Ahamed, Zheng Shilong, Wang Guangdi

SAT-341 Pharmacology and Metabolism of GLL398 an Oral Selective Estrogen Receptor Degrader for Endocrine Therapy of Breast Cancer

SAT-341:GLL398(一种用于乳腺癌内分泌治疗的口服选择性雌激素受体降解剂)的药理学和代谢

Tiwari, Anshuly; Modi, Siddharth J; Girme, Aboli; Hingorani, Lal; Guo, Shanchun; Hossain, Ahamed; Zhang, Changde; Mottamal, Madhu; Liu, Jiawang; Wiese, Thomas; Wang, Guangdi

Point-of-Care Determination of Acetaminophen Levels with Multi-Hydrogen Bond Manipulated Single-Molecule Recognition (eMuHSiR)

利用多氢键操纵的单分子识别技术(eMuHSiR)即时测定对乙酰氨基酚水平

Zhang, Yan; Huang, Zhongyuan; Wang, Letao; Wang, Chunming; Zhang, Changde; Wiese, Tomas; Wang, Guangdi; Riley, Kevin; Wang, Zhe

Structure-activity relationship and pharmacokinetic studies of 3-O-substitutedflavonols as anti-prostate cancer agents

3-O-取代黄酮醇作为抗前列腺癌药物的构效关系和药代动力学研究

Li, Xiang; Zhang, Changde; Guo, Shanchun; Rajaram, Pravien; Lee, Maizie; Chen, Guanglin; Fong, Ryan; Gonzalez, Aaron; Zhang, Qiang; Zheng, Shilong; Wang, Guangdi; Chen, Qiao-Hong

Structure-Activity Relationship and Pharmacokinetic Studies of 1,5-Diheteroarylpenta-1,4-dien-3-ones: A Class of Promising Curcumin-Based Anticancer Agents

1,5-二杂芳基戊-1,4-二烯-3-酮的构效关系及药代动力学研究:一类有前景的姜黄素类抗癌药物

Rubing Wang, Chengsheng Chen, Xiaojie Zhang, Changde Zhang, Qiu Zhong, Guanglin Chen, Qiang Zhang, Shilong Zheng, Guangdi Wang, Qiao-Hong Chen

Boronic prodrug of endoxifen as an effective hormone therapy for breast cancer

硼酸前药内多昔芬作为一种有效的乳腺癌激素疗法

Zhang, Changde; Zhong, Qiu; Zhang, Qiang; Zheng, Shilong; Miele, Lucio; Wang, Guangdi

Novel aspirin-triggered neuroprotectin D1 attenuates cerebral ischemic injury after experimental stroke

新型阿司匹林触发的神经保护素D1可减轻实验性卒中后的脑缺血损伤。

Bazan, Nicolas G; Eady, Tiffany N; Khoutorova, Larissa; Atkins, Kristal D; Hong, Song; Lu, Yan; Zhang, Changde; Jun, Bokkyoo; Obenaus, Andre; Fredman, Gabrielle; Zhu, Min; Winkler, Jeremy W; Petasis, Nicos A; Serhan, Charles N; Belayev, Ludmila

Docosahexaenoic acid signaling modulates cell survival in experimental ischemic stroke penumbra and initiates long-term repair in young and aged rats.

二十二碳六烯酸信号传导调节实验性缺血性中风半暗带中的细胞存活,并启动年轻和老年大鼠的长期修复

Eady Tiffany N, Belayev Ludmila, Khoutorova Larissa, Atkins Kristal D, Zhang Changde, Bazan Nicolas G

Lipid-mediated cell signaling protects against injury and neurodegeneration

脂质介导的细胞信号传导可抵抗损伤和神经退行性变

Zhang, Changde; Bazan, Nicolas G