Design of N-Benzoxaborole Benzofuran GSK8175-Optimization of Human Pharmacokinetics Inspired by Metabolites of a Failed Clinical HCV Inhibitor
受失败的临床HCV抑制剂代谢产物启发,设计N-苯并噁硼杂环苯并呋喃GSK8175——优化人体药代动力学
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.8b01719
Chong, Pek Y; Shotwell, J Brad; Miller, John; Price, Daniel J; Maynard, Andy; Voitenleitner, Christian; Mathis, Amanda; Williams, Shawn; Pouliot, Jeffrey J; Creech, Katrina; Wang, Feng; Fang, Jing; Zhang, Huichang; Tai, Vincent W-F; Turner, Elizabeth; Kahler, Kirsten M; Crosby, Renae; Peat, Andrew J