Chemical remodeling of a cellular chaperone to target the active state of mutant KRAS
通过化学方法改造细胞伴侣蛋白,使其靶向突变型KRAS的活性状态
期刊:Science
影响因子:45.8
doi:10.1126/science.adg9652
Schulze, Christopher J; Seamon, Kyle J; Zhao, Yulei; Yang, Yu C; Cregg, Jim; Kim, Dongsung; Tomlinson, Aidan; Choy, Tiffany J; Wang, Zhican; Sang, Ben; Pourfarjam, Yasin; Lucas, Jessica; Cuevas-Navarro, Antonio; Ayala-Santos, Carlos; Vides, Alberto; Li, Chuanchuan; Marquez, Abby; Zhong, Mengqi; Vemulapalli, Vidyasiri; Weller, Caroline; Gould, Andrea; Whalen, Daniel M; Salvador, Anthony; Milin, Anthony; Saldajeno-Concar, Mae; Dinglasan, Nuntana; Chen, Anqi; Evans, Jim; Knox, John E; Koltun, Elena S; Singh, Mallika; Nichols, Robert; Wildes, David; Gill, Adrian L; Smith, Jacqueline A M; Lito, Piro