Development of a brain-penetrant G9a methylase inhibitor to target Alzheimer's disease-associated proteopathology.
开发一种可穿透血脑屏障的 G9a 甲基化酶抑制剂,以靶向治疗阿尔茨海默病相关的蛋白质病理
期刊:Nature Communications
影响因子:15.7
doi:10.1038/s41467-025-59128-z
Xie Ling, Sheehy Ryan N, Muneer Adil, Xiong Yan, Wrobel John A, Zhang Feng, Park Kwang-Su, Velez Julia, Liu Jing, Luo Yan-Jia, Asrican Brent, Dong Ping, Li Ya-Dong, Damian Corina, Quintanilla Luis, Li Yongyi, Xu Chongchong, Deshmukh Mohanish, Coleman Leon G Jr, Ming Guo-Li, Song Hongjun, Wen Zhexing, Jin Jian, Song Juan, Chen Xian