日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Glucose metabolism controls oxidative burst and lipid mediator production in neutrophils upon microbial challenge

葡萄糖代谢控制中性粒细胞在受到微生物攻击时的氧化爆发和脂质介质生成。

Freitag, Alexandra; Günther, Kerstin; Campillo Prados, Miriam; Hochrein, Sophia M; Schmitz, Werner; Sinning, Katrin; Zischinsky, Gunther; Klebl, Bert; Ohlsen, Knut; Morschhäuser, Joachim; Werz, Oliver; Jordan, Paul M; Vaeth, Martin

Avapritinib-based SAR studies unveil a binding pocket in KIT and PDGFRA

基于 Avapritinib 的 SAR 研究揭示了 KIT 和 PDGFRA 中的结合位点

A Teuber #, T Schulz #, B S Fletcher, R Gontla, T Mühlenberg, M-L Zischinsky, J Niggenaber, J Weisner, S B Kleinbölting, J Lategahn, S Sievers, M P Müller, S Bauer, D Rauh

Inhibiting the glycerophosphodiesterase EDI3 in ER-HER2+ breast cancer cells resistant to HER2-targeted therapy reduces viability and tumour growth

抑制对 HER2 靶向治疗有抗性的 ER-HER2+ 乳腺癌细胞中的甘油磷酸二酯酶 EDI3 可降低细胞活力和肿瘤生长

Magdalena Keller #, Katharina Rohlf #, Annika Glotzbach #, Gregor Leonhardt, Simon Lüke, Katharina Derksen, Özlem Demirci, Defne Göçener, Mohammad AlWahsh, Jörg Lambert, Cecilia Lindskog, Marcus Schmidt, Walburgis Brenner, Matthias Baumann, Eldar Zent, Mia-Lisa Zischinsky, Birte Hellwig, Katrin Madj

The Pseudo-Natural Product Rhonin Targets RHOGDI

伪天然产物罗宁靶向RHOGDI

Akbarzadeh, Mohammad; Flegel, Jana; Patil, Sumersing; Shang, Erchang; Narayan, Rishikesh; Buchholzer, Marcel; Kazemein Jasemi, Neda S; Grigalunas, Michael; Krzyzanowski, Adrian; Abegg, Daniel; Shuster, Anton; Potowski, Marco; Karatas, Hacer; Karageorgis, George; Mosaddeghzadeh, Niloufar; Zischinsky, Mia-Lisa; Merten, Christian; Golz, Christopher; Brieger, Lucas; Strohmann, Carsten; Antonchick, Andrey P; Janning, Petra; Adibekian, Alexander; Goody, Roger S; Ahmadian, Mohammad Reza; Ziegler, Slava; Waldmann, Herbert

Dual Inhibition of GSK3β and CDK5 Protects the Cytoskeleton of Neurons from Neuroinflammatory-Mediated Degeneration In Vitro and In Vivo

双重抑制GSK3β和CDK5可在体外和体内保护神经元细胞骨架免受神经炎症介导的退行性变。

Reinhardt, Lydia; Kordes, Susanne; Reinhardt, Peter; Glatza, Michael; Baumann, Matthias; Drexler, Hannes C A; Menninger, Sascha; Zischinsky, Gunther; Eickhoff, Jan; Fröb, Claudia; Bhattarai, Prabesh; Arulmozhivarman, Guruchandar; Marrone, Lara; Janosch, Antje; Adachi, Kenjiro; Stehling, Martin; Anderson, Eric N; Abo-Rady, Masin; Bickle, Marc; Pandey, Udai Bhan; Reimer, Michell M; Kizil, Caghan; Schöler, Hans R; Nussbaumer, Peter; Klebl, Bert; Sterneckert, Jared L

Dynarrestin, a Novel Inhibitor of Cytoplasmic Dynein

Dynarrestin,一种新型细胞质动力蛋白抑制剂

Susanne Höing, Ting-Yu Yeh, Matthias Baumann, Nancy E Martinez, Peter Habenberger, Lea Kremer, Hannes C A Drexler, Philipp Küchler, Peter Reinhardt, Axel Choidas, Mia-Lisa Zischinsky, Gunther Zischinsky, Swaran Nandini, Aaron P Ledray, Stephanie A Ketcham, Lydia Reinhardt, Masin Abo-Rady, Michael Gl

A novel CDK7 inhibitor of the Pyrazolotriazine class exerts broad-spectrum antiviral activity at nanomolar concentrations

吡唑并三嗪类新型 CDK7 抑制剂在纳摩尔浓度下发挥广谱抗病毒活性

Corina Hutterer, Jan Eickhoff, Jens Milbradt, Klaus Korn, Isabel Zeitträger, Hanife Bahsi, Sabrina Wagner, Gunther Zischinsky, Alexander Wolf, Carsten Degenhart, Anke Unger, Matthias Baumann, Bert Klebl, Manfred Marschall

alpha5beta1 Integrin blockade inhibits lymphangiogenesis in airway inflammation

α5β1整合素阻断可抑制气道炎症中的淋巴管生成

Okazaki, Tatsuma; Ni, Amy; Ayeni, Oluwasheyi A; Baluk, Peter; Yao, Li-Chin; Vossmeyer, Doerte; Zischinsky, Gunther; Zahn, Grit; Knolle, Jochen; Christner, Claudia; McDonald, Donald M