日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Synthesis, Computational Studies, and Structural Analysis of 1-(3,5-Dimethoxyphenyl)azetidin-2-ones with Antiproliferative Activity in Breast Cancer and Chemoresistant Colon Cancer

1-(3,5-二甲氧基苯基)氮杂环丁酮类化合物的合成、计算研究及结构分析及其在乳腺癌和化疗耐药性结肠癌中的抗增殖活性

Malebari, Azizah M; Kandwal, Shubhangi; Ali, Abdirahman; Fayne, Darren; Twamley, Brendan; Zisterer, Daniela M; Meegan, Mary J

Correction: Wang et al. Antiproliferative and Tubulin-Destabilising Effects of 3-(Prop-1-en-2-yl)azetidin-2-Ones and Related Compounds in MCF-7 and MDA-MB-231 Breast Cancer Cells. Pharmaceuticals 2023, 16, 1000

更正:Wang 等人,《3-(丙-1-烯-2-基)氮杂环丁酮及其相关化合物对 MCF-7 和 MDA-MB-231 乳腺癌细胞的抗增殖和微管蛋白去稳定作用》,Pharmaceuticals 2023, 16, 1000

Wang, Shu; Malebari, Azizah M; Greene, Thomas F; Kandwal, Shubhangi; Fayne, Darren; Nathwani, Seema M; Zisterer, Daniela M; Twamley, Brendan; O'Boyle, Niamh M; Meegan, Mary J

Correction: Malebari et al. Synthesis and Antiproliferative Evaluation of 3-Chloroazetidin-2-ones with Antimitotic Activity: Heterocyclic Bridged Analogues of Combretastatin A-4. Pharmaceuticals 2021, 14, 1119

更正:Malebari 等人,《具有抗有丝分裂活性的 3-氯氮杂环丁酮-2-酮的合成及抗增殖评价:康布瑞他汀 A-4 的杂环桥联类似物》,Pharmaceuticals 2021, 14, 1119

Malebari, Azizah M; Wang, Shu; Greene, Thomas F; O'Boyle, Niamh M; Fayne, Darren; Khan, Mohemmed Faraz; Nathwani, Seema M; Twamley, Brendan; McCabe, Thomas; Zisterer, Daniela M; Meegan, Mary J

Probing the metalloproteome: an 8-mercaptoquinoline motif enriches minichromosome maintenance complex components as significant metalloprotein targets in live cells

金属蛋白组学研究:8-巯基喹啉基序富集微染色体维持复合物组分,使其成为活细胞中重要的金属蛋白靶点

McKenna, Sean M; Florea, Bogdan I; Zisterer, Daniela M; van Kasteren, Sander I; McGouran, Joanna F

The role of the Nrf2/GSH antioxidant system in cisplatin resistance in malignant rhabdoid tumours

Nrf2/GSH 抗氧化系统在恶性横纹肌瘤顺铂耐药中的作用

Patricia Hannon Barroeta, Maureen J O'Sullivan, Daniela M Zisterer

Antiproliferative and Tubulin-Destabilising Effects of 3-(Prop-1-en-2-yl)azetidin-2-Ones and Related Compounds in MCF-7 and MDA-MB-231 Breast Cancer Cells

3-(丙-1-烯-2-基)氮杂环丁-2-酮及其相关化合物对 MCF-7 和 MDA-MB-231 乳腺癌细胞的抗增殖和微管蛋白不稳定作用

Shu Wang, Azizah M Malebari, Thomas F Greene, Shubhangi Kandwal, Darren Fayne, Seema M Nathwani, Daniela M Zisterer, Brendan Twamley, Niamh M O'Boyle, Mary J Meegan

Synthesis, Characterisation and Mechanism of Action of Anticancer 3-Fluoroazetidin-2-ones

抗癌化合物3-氟氮杂环丁酮的合成、表征及作用机制

Malebari, Azizah M; Duffy Morales, Gabriela; Twamley, Brendan; Fayne, Darren; Khan, Mohemmed Faraz; McLoughlin, Eavan C; O'Boyle, Niamh M; Zisterer, Daniela M; Meegan, Mary J

Identification of Src as a Therapeutic Target in Oesophageal Adenocarcinoma through Functional Genomic and High-Throughput Drug Screening Approaches

通过功能基因组和高通量药物筛选方法鉴定 Src 作为食管腺癌的治疗靶点

Niamh H McCabe, Leanne Stevenson, Enya Scanlon, Rosalie Douglas, Susanna Kennedy, Oliver Keminer, Björn Windshügel, Daniela Zisterer, Richard D Kennedy, Jaine K Blayney, Richard C Turkington

Synthesis and Biological Evaluation of 1-(Diarylmethyl)-1 H-1,2,4-triazoles and 1-(Diarylmethyl)-1 H-imidazoles as a Novel Class of Anti-Mitotic Agent for Activity in Breast Cancer

1-(二芳甲基)-1 H-1,2,4-三唑和 1-(二芳甲基)-1 H-咪唑作为新型抗有丝分裂剂对乳腺癌的活性合成及生物学评价

Gloria Ana, Patrick M Kelly, Azizah M Malebari, Sara Noorani, Seema M Nathwani, Brendan Twamley, Darren Fayne, Niamh M O'Boyle, Daniela M Zisterer, Elisangela Flavia Pimentel, Denise Coutinho Endringer, Mary J Meegan

Synthesis and Antiproliferative Evaluation of 3-Chloroazetidin-2-ones with Antimitotic Activity: Heterocyclic Bridged Analogues of Combretastatin A-4

具有抗有丝分裂活性的 3-氯氮杂环丁烷-2-酮的合成及抗增殖评价:Combretastatin A-4 的杂环桥接类似物

Azizah M Malebari, Shu Wang, Thomas F Greene, Niamh M O'Boyle, Darren Fayne, Mohemmed Faraz Khan, Seema M Nathwani, Brendan Twamley, Thomas McCabe, Daniela M Zisterer, Mary J Meegan