日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Design and Synthesis of Caffeine-Based Derivatives with Antioxidant and Neuroprotective Activity: In Vitro Evaluation and SwissADME Profiling

具有抗氧化和神经保护活性的咖啡因衍生物的设计与合成:体外评价和SwissADME分析

Stefanova, Denitsa; Garip, Alime; Tzankova, Virginia; Kostov, Stefan; Mateev, Emilio; Zlatkov, Alexander; Mitkov, Yavor

Activating FGFR1 restores Integrin-β1-mediated fibronectin sensing in satellite cells of aged mice.

激活 FGFR1 可恢复老年小鼠卫星细胞中整合素-β1 介导的纤连蛋白感知。

Chang Tze-Ling, Vallery Tenaya K, Zlatkov Thea S, Cutler Alicia A, Kurland Jesse V, Butcher Carson H, Anseth Kristi S, Olwin Bradley B

Sublytic Activity of a Pore-Forming Protein From Commensal Bacteria Causes Epigenetic Modulation of Tumour-Affiliated Protein Expression.

共生细菌中成孔蛋白的亚溶血活性导致肿瘤相关蛋白表达的表观遗传调控

Toh Eric, Baryalai Palwasha, Nadeem Aftab, Aung Kyaw Min, Myint Si Lhyam, Zlatkov Nikola, Alidadi Hadis, Zhu Shaochun, Mateus André, Raina Deepak Bushan, Ramstedt Madeleine, Uhlin Bernt Eric, Wai Sun Nyunt

A new understanding of Acanthamoeba castellanii: dispelling the role of bacterial pore-forming toxins in cyst formation and amoebicidal actions.

对棘阿米巴属卡氏阿米巴的新认识:揭穿细菌成孔毒素在包囊形成和杀阿米巴作用中的作用

Yabrag Abdelbasset, Ullah Naeem, Baryalai Palwasha, Ahmad Irfan, Zlatkov Nikola, Toh Eric, Lindbäck Toril, Uhlin Bernt Eric, Wai Sun Nyunt, Nadeem Aftab

Design, Synthesis, and Evaluation of Pyrrole-Based Selective MAO-B Inhibitors with Additional AChE Inhibitory and Neuroprotective Properties Identified via Virtual Screening

通过虚拟筛选鉴定出具有额外AChE抑制和神经保护特性的吡咯基选择性MAO-B抑制剂的设计、合成和评价

Mateev, Emilio; Chtita, Samir; Pavlova, Ekaterina; Irfan, Ali; Tzankova, Diana; Sharma, Shubham; Georgiev, Borislav; Mateeva, Alexandrina; Momekov, Georgi; Georgieva, Maya; Zlatkov, Alexander; Kondeva-Burdina, Magdalena

Classical Paal-Knorr Cyclization for Synthesis of Pyrrole-Based Aryl Hydrazones and In Vitro/In Vivo Evaluation on Pharmacological Models of Parkinson's Disease

经典的Paal-Knorr环化反应用于合成吡咯基芳基腙及其在帕金森病药理模型中的体外/体内评价

Georgieva, Maya; Sharkov, Martin; Mateev, Emilio; Tzankova, Diana; Popov, Georgi; Manov, Vasil; Zlatkov, Alexander; Simeonova, Rumyana; Kondeva-Burdina, Magdalena

Cardiopulmonary Reactivity in Bulgarian National Taekwon-Do Team Athletes

保加利亚国家跆拳道队运动员的心肺反应性

Zlatkova, Krasimira; Zlatkov, Yuliyan; Kostova, Radostina

Neurotoxicity, Neuroprotection, In Vitro MAOA/MAOB Inhibitory Activity Assessment, Molecular Docking, and Permeability Assay Studies of Newly Synthesized Hydrazones Containing a Pyrrole Ring

对新合成的含吡咯环的腙类化合物进行神经毒性、神经保护、体外MAOA/MAOB抑制活性评估、分子对接和渗透性测定研究

Georgieva, Maya; Mateev, Emilio; Valkova, Iva; Kuteva, Hristina; Tzankova, Diana; Stefanova, Denitsa; Yordanov, Yordan; Lybomirova, Karolina; Zlatkov, Alexander; Tzankova, Virginia; Kondeva-Burdina, Magdalena

In Silico and Chromatographic Methods for Analysis of Biotransformation of Prospective Neuroprotective Pyrrole-Based Hydrazone in Isolated Rat Hepatocytes

利用计算机模拟和色谱法分析潜在神经保护性吡咯基腙在分离的大鼠肝细胞中的生物转化

Mateeva, Alexandrina; Kondeva-Burdina, Magdalena; Mateev, Emilio; Nedialkov, Paraskev; Lyubomirova, Karolina; Peikova, Lily; Georgieva, Maya; Zlatkov, Alexander

The adsorption of drugs on nanoplastics has severe biological impact

药物在纳米塑料上的吸附会对生物体产生严重影响。

Dick, Leonard; Batista, Patrick R; Zaby, Paul; Manhart, Gabriele; Kopatz, Verena; Kogler, Lukas; Pichler, Verena; Grebien, Florian; Bakos, Vince; Plósz, Benedek G; Kolev, Nikola Zlatkov; Kenner, Lukas; Kirchner, Barbara; Hollóczki, Oldamur