Structure-guided design of 7-azaindole DNMT1 inhibitors active against hypomethylating agent-resistant acute myeloid leukemia
基于结构的7-氮杂吲哚DNMT1抑制剂设计,可有效对抗低甲基化药物耐药的急性髓系白血病
期刊:Proceedings of the National Academy of Sciences of the United States of America
影响因子:9.1
doi:10.1073/pnas.2532472123
Tang, Shibing; Zong, Liangyi; Ma, Shuyuan; Shang, Yini; Wei, Jiale; Liu, Jianguang; Cui, Ying; Guo, Huahui; Zou, Kang; Wang, Kezhi; Li, Hongkun; Ye, Fei; Huang, Jing; Luo, Cheng; Li, Zhihai; Baylin, Stephen B; Kong, Xiangqian