Stapled Peptides as HIF-1α/p300 Inhibitors: Helicity Enhancement in the Bound State Increases Inhibitory Potency
钉合肽作为 HIF-1α/p300 抑制剂:结合状态下螺旋度增强可提高抑制效力
期刊:Chemistry
影响因子:2.4
doi:10.1002/chem.202000417
Kristina Hetherington, Zsofia Hegedus, Thomas A Edwards, Richard B Sessions, Adam Nelson, Andrew J Wilson