A Chemical Probe for Dark Kinase STK17B Derives Its Potency and High Selectivity through a Unique P-Loop Conformation.
一种用于暗激酶 STK17B 的化学探针,其高效性和高选择性源于其独特的 P 环构象
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.0c01174
Picado Alfredo, Chaikuad Apirat, Wells Carrow I, Shrestha Safal, Zuercher William J, Pickett Julie E, Kwarcinski Frank E, Sinha Parvathi, de Silva Chandi S, Zutshi Reena, Liu Shubin, Kannan Natarajan, Knapp Stefan, Drewry David H, Willson Timothy M