日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Disconnect between in vitro and in vivo efficacy of the MPS1 inhibitor NTRC 0066-0 against glioblastoma

MPS1抑制剂NTRC 0066-0在体外和体内抗胶质母细胞瘤疗效上的差异

de Gooijer, Mark C; Fedorushkova, Daria M; Zhang, Ping; Buil, Levi C M; Çitirikkaya, Ceren H; Çolakoğlu, Hilal; Maia, Ana Rita R; Bočkaj, Irena; Espitia-Ballestas, Margarita; Kuil, Laura E; Beijnen, Jos H; van Tellingen, Olaf

Reanalysis of in vivo drug synergy validation study rules out synergy in most cases

对体内药物协同作用验证研究的重新分析排除了大多数情况下的协同作用。

van Tellingen, Olaf; de Menezes, Renee X

Cranial radiotherapy profoundly affects glia without inducing widespread cellular senescence

颅脑放射治疗对神经胶质细胞有显著影响,但不会诱发广泛的细胞衰老。

Kuil, Laura E; van Scheppingen, Roan H; Leter, Yoran M; Röring, Berend H; de Gooijer, Mark C; van Heijningen, Caroline L; Prekovic, Stefan; Compter, Annette; van Tellingen, Olaf; Schagen, Sanne B

EXTH-118. Development of a multi-target drug combination targeting three major proliferation pathways in glioblastoma

EXTH-118. 开发一种针对胶质母细胞瘤三大主要增殖通路的多靶点药物组合

Wang, F; Xue, X; Wei, J; An, Y; Yao, J; Cai, H; Wu, J; Dai, C; Qian, Z; Xu, Z; Miao, Y; Their, Anna; Elens, Robert; Baltira, Chrysiida; Szewczyk, Aldona; Rozing, Kicky; Beijnen, Jos; de Gooijer, Mark; van Tellingen, Olaf

A pharmacokinetic study and critical reappraisal of curcumin formulations enhancing bioavailability

一项药代动力学研究和对提高生物利用度的姜黄素制剂的重新评价

Kroon, Maurice A G M; van Laarhoven, Hanneke W M; Swart, Eleonora L; van Tellingen, Olaf; Kemper, E Marleen

The impact of ATP-binding cassette transporters in the diseased brain: Context matters

ATP结合盒转运蛋白在病变大脑中的作用:背景因素很重要

Baltira, Chrysiida; Aronica, Eleonora; Elmquist, William F; Langer, Oliver; Löscher, Wolfgang; Sarkaria, Jann N; Wesseling, Pieter; de Gooijer, Mark C; van Tellingen, Olaf

Non-therapeutic plasma levels in individuals utilizing curcumin supplements in daily life

日常生活中服用姜黄素补充剂的个体血浆中姜黄素水平低于治疗水平

Kroon, Maurice A G M; Berbee, Jacqueline K; Majait, Soumia; Swart, Eleonora L; van Tellingen, Olaf; van Laarhoven, Hanneke W M; Kemper, E Marleen

Author Correction: Tryptophan depletion results in tryptophan-to-phenylalanine substitutants

作者更正:色氨酸耗竭导致色氨酸被苯丙氨酸取代。

Pataskar, Abhijeet; Champagne, Julien; Nagel, Remco; Kenski, Juliana; Laos, Maarja; Michaux, Justine; Pak, Hui Song; Bleijerveld, Onno B; Mordente, Kelly; Navarro, Jasmine Montenegro; Blommaert, Naomi; Nielsen, Morten M; Lovecchio, Domenica; Stone, Everett; Georgiou, George; de Gooijer, Mark C; van Tellingen, Olaf; Altelaar, Maarten; Joosten, Robbie P; Perrakis, Anastassis; Olweus, Johanna; Bassani-Sternberg, Michal; Peeper, Daniel S; Agami, Reuven

Comments on: "Synergistic activity of mTORC1/2 kinase and MEK inhibitors suppresses pediatric low-grade glioma tumorigenicity and vascularity"

关于“mTORC1/2激酶和MEK抑制剂的协同作用抑制儿童低级别胶质瘤的致瘤性和血管生成”的评论

van Tellingen, Olaf; de Gooijer, Mark C; Sarkaria, Jann N; Elmquist, William F

Expression and Cellular Distribution of P-Glycoprotein and Breast Cancer Resistance Protein in Amyotrophic Lateral Sclerosis Patients

肌萎缩侧索硬化症患者中P-糖蛋白和乳腺癌抗性蛋白的表达及细胞分布

van Vliet, Erwin A; Iyer, Anand M; Mesarosova, Lucia; Çolakoglu, Hilal; Anink, Jasper J; van Tellingen, Olaf; Maragakis, Nicholas J; Shefner, Jeremy; Bunt, Ton; Aronica, Eleonora