日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The endocannabinoid 2-arachidonoylglycerol is released and transported on demand via extracellular microvesicles.

内源性大麻素 2-花生四烯酸甘油酯可按需通过细胞外微囊泡释放和运输

Straub Verena M, Barti Benjamin, Tandar Sebastian T, Stevens A Floor, van Egmond Noëlle, van der Wel Tom, Zhu Na, Rüegger Joel, van der Horst Cas, Heitman Laura H, Li Yulong, Stella Nephi, van Hasselt J G Coen, Katona István, van der Stelt Mario

Comparative Photoaffinity Profiling of Omega-3 Signaling Lipid Probes Reveals Prostaglandin Reductase 1 as a Metabolic Hub in Human Macrophages

ω-3信号脂质探针的光亲和力比较分析揭示前列腺素还原酶1是人类巨噬细胞中的代谢枢纽

Gagestein, Berend; von Hegedus, Johannes H; Kwekkeboom, Joanneke C; Heijink, Marieke; Blomberg, Niek; van der Wel, Tom; Florea, Bogdan I; van den Elst, Hans; Wals, Kim; Overkleeft, Herman S; Giera, Martin; Toes, René E M; Ioan-Facsinay, Andreea; van der Stelt, Mario

Detection of cannabinoid receptor type 2 in native cells and zebrafish with a highly potent, cell-permeable fluorescent probe

利用高效、细胞渗透性荧光探针检测天然细胞和斑马鱼中的大麻素受体2型

Gazzi, Thais; Brennecke, Benjamin; Atz, Kenneth; Korn, Claudia; Sykes, David; Forn-Cuni, Gabriel; Pfaff, Patrick; Sarott, Roman C; Westphal, Matthias V; Mostinski, Yelena; Mach, Leonard; Wasinska-Kalwa, Malgorzata; Weise, Marie; Hoare, Bradley L; Miljuš, Tamara; Mexi, Maira; Roth, Nicolas; Koers, Eline J; Guba, Wolfgang; Alker, André; Rufer, Arne C; Kusznir, Eric A; Huber, Sylwia; Raposo, Catarina; Zirwes, Elisabeth A; Osterwald, Anja; Pavlovic, Anto; Moes, Svenja; Beck, Jennifer; Nettekoven, Matthias; Benito-Cuesta, Irene; Grande, Teresa; Drawnel, Faye; Widmer, Gabriella; Holzer, Daniela; van der Wel, Tom; Mandhair, Harpreet; Honer, Michael; Fingerle, Jürgen; Scheffel, Jörg; Broichhagen, Johannes; Gawrisch, Klaus; Romero, Julián; Hillard, Cecilia J; Varga, Zoltan V; van der Stelt, Mario; Pacher, Pal; Gertsch, Jürg; Ullmer, Christoph; McCormick, Peter J; Oddi, Sergio; Spaink, Herman P; Maccarrone, Mauro; Veprintsev, Dmitry B; Carreira, Erick M; Grether, Uwe; Nazaré, Marc

Activity-based protein profiling reveals off-target proteins of the FAAH inhibitor BIA 10-2474

基于活性的蛋白质谱分析揭示了FAAH抑制剂BIA 10-2474的脱靶蛋白

van Esbroeck, Annelot C M; Janssen, Antonius P A; Cognetta, Armand B 3rd; Ogasawara, Daisuke; Shpak, Guy; van der Kroeg, Mark; Kantae, Vasudev; Baggelaar, Marc P; de Vrij, Femke M S; Deng, Hui; Allarà, Marco; Fezza, Filomena; Lin, Zhanmin; van der Wel, Tom; Soethoudt, Marjolein; Mock, Elliot D; den Dulk, Hans; Baak, Ilse L; Florea, Bogdan I; Hendriks, Giel; De Petrocellis, Luciano; Overkleeft, Herman S; Hankemeier, Thomas; De Zeeuw, Chris I; Di Marzo, Vincenzo; Maccarrone, Mauro; Cravatt, Benjamin F; Kushner, Steven A; van der Stelt, Mario

Chiral disubstituted piperidinyl ureas: a class of dual diacylglycerol lipase-α and ABHD6 inhibitors

手性二取代哌啶基脲:一类双重二酰甘油脂肪酶-α和ABHD6抑制剂

Deng, Hui; van der Wel, Tom; van den Berg, Richard J B H N; van den Nieuwendijk, Adrianus M C H; Janssen, Freek J; Baggelaar, Marc P; Overkleeft, Hermen S; van der Stelt, Mario

Highly Selective, Reversible Inhibitor Identified by Comparative Chemoproteomics Modulates Diacylglycerol Lipase Activity in Neurons

通过比较化学蛋白质组学鉴定出的高选择性、可逆抑制剂可调节神经元中的二酰甘油脂肪酶活性

Baggelaar, Marc P; Chameau, Pascal J P; Kantae, Vasudev; Hummel, Jessica; Hsu, Ku-Lung; Janssen, Freek; van der Wel, Tom; Soethoudt, Marjolein; Deng, Hui; den Dulk, Hans; Allarà, Marco; Florea, Bogdan I; Di Marzo, Vincenzo; Wadman, Wytse J; Kruse, Chris G; Overkleeft, Herman S; Hankemeier, Thomas; Werkman, Taco R; Cravatt, Benjamin F; van der Stelt, Mario