日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Shaping Antimalarials: A Geometry-First Approach to PfCLK3 Covalent Inhibitors

抗疟药的调控:一种基于几何结构的PfCLK3共价抑制剂设计方法

Brettell, Skye B; Fuentes-Guerra Bustos, Carla; Sharma, Saumya; Cann, Gillian; Carruthers, Lauren V; Begen, Abbey; Milligan, Graeme; Clarke, David J; Tobin, Andrew B; Jamieson, Andrew G

Oncogenic DEAD-box ATPase DDX41 establishes transcript ensembles via CLK3-dependent and -independent mechanisms

致癌性DEAD-box ATPase DDX41通过CLK3依赖性和非依赖性机制建立转录本集合。

Jeong-Ah Kim # ,Siqi Shen # ,Christina M Jurotich ,Saritha S D'Souza ,Johnathan J Caldon ,Igor I Slukvin ,Jane E Churpek ,Sunduz Keles ,Emery H Bresnick

Deciphering the unique autoregulatory mechanisms and substrate specificity of the understudied DCLK3 kinase linked to neurodegenerative diseases

解析与神经退行性疾病相关的、研究不足的DCLK3激酶独特的自调节机制和底物特异性

Lu, Jason D; Zhao, Peng; Prasad, Anup; Gupta, Neha; Gravel, Nathan; Shidhaye, Tej; Wells, Lance; Katiyar, Samiksha; Kannan, Natarajan

Lysine targeting covalent inhibitors of malarial kinase PfCLK3

赖氨酸靶向共价抑制疟原虫激酶 PfCLK3 的抑制剂

Brettell, Skye B; Cann, Gillian; Begen, Abbey; Sharma, Saumya; Mahindra, Amit; Carruthers, Lauren V; Milligan, Graeme; Clarke, David J; Tobin, Andrew B; Jamieson, Andrew G

Research towards selective inhibition of the CLK3 kinase

针对CLK3激酶选择性抑制的研究

Singh, Vinay Kumar; Justaud, Frédéric; Brahmaiah, Dabbugoddu; Kumar, Nangunoori Sampath; Baratte, Blandine; Robert, Thomas; Bach, Stéphane; Reddy, Chada Raji; Levoin, Nicolas; Grée, René L

Targeting PfCLK3 with Covalent Inhibitors: A Novel Strategy for Malaria Treatment

利用共价抑制剂靶向 PfCLK3:一种治疗疟疾的新策略

Brettell, Skye B; Janha, Omar; Begen, Abbey; Cann, Gillian; Sharma, Saumya; Olaniyan, Niniola; Yelland, Tamas; Hole, Alison J; Alam, Benazir; Mayville, Emily; Gillespie, Ross; Capper, Michael; Fidock, David A; Milligan, Graeme; Clarke, David J; Tobin, Andrew B; Jamieson, Andrew G

Retraction: MiR-1236-3p inhibits the proliferation, invasion, and migration of colon cancer cells and hinders epithelial-mesenchymal transition by targeting DCLK3

撤稿:miR-1236-3p通过靶向DCLK3抑制结肠癌细胞的增殖、侵袭和迁移,并阻碍上皮-间质转化。

A CLK3-HMGA2 Alternative Splicing Axis Impacts Human Hematopoietic Stem Cell Molecular Identity throughout Development

CLK3-HMGA2选择性剪接轴在发育过程中影响人类造血干细胞的分子特性

Marcella Cesana ,Michael H Guo ,Davide Cacchiarelli ,Lara Wahlster ,Jessica Barragan ,Sergei Doulatov ,Linda T Vo ,Beatrice Salvatori ,Cole Trapnell ,Kendell Clement ,Patrick Cahan ,Kaloyan M Tsanov ,Patricia M Sousa ,Barbara Tazon-Vega ,Adriano Bolondi ,Federico M Giorgi ,Andrea Califano ,John L Rinn ,Alexander Meissner ,Joel N Hirschhorn ,George Q Daley

CLK-dependent exon recognition and conjoined gene formation revealed with a novel small molecule inhibitor

新型小分子抑制剂揭示 CLK 依赖的外显子识别和连体基因形成

Tyler Funnell, Shinya Tasaki, Arusha Oloumi, Shinsuke Araki, Esther Kong, Damian Yap, Yusuke Nakayama, Christopher S Hughes, S-W Grace Cheng, Hirokazu Tozaki, Misa Iwatani, Satoshi Sasaki, Tomohiro Ohashi, Tohru Miyazaki, Nao Morishita, Daisuke Morishita, Mari Ogasawara-Shimizu, Momoko Ohori, Shoich