日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Molecular dynamics simulations elucidate the role of the F-F' loop in substrate entry into CYP3A4

分子动力学模拟阐明了FF'环在底物进入CYP3A4中的作用

Yan, Junfang; Hirao, Hajime

Repeated Intake of Grapefruit Juice Inhibits CYP2B6, CYP2C9, CYP2C19, and CYP3A4 while Lingonberry Powder Does Not Induce Major CYP Enzymes in Humans

反复摄入葡萄柚汁会抑制CYP2B6、CYP2C9、CYP2C19和CYP3A4,而越橘粉不会诱导人体内主要的CYP酶。

Aurinsalo, Laura; Lapatto-Reiniluoto, Outi; Kurkela, Mika; Neuvonen, Mikko; Moilanen, Eeva; Niemi, Mikko; Tornio, Aleksi; Backman, Janne T

LRRC8A Inhibition Overcomes Chemoresistance by Downregulating MRP3 and CYP3A4 in the 3D Spheroid Model of Human Breast Cancer Cells.

LRRC8A 抑制剂通过下调 3D 球状体模型中 MRP3 和 CYP3A4 来克服人类乳腺癌细胞的化疗耐药性。

Otsuka Ryo, Kajikuri Junko, Matsui Miki, Kito Hiroaki, Kitahara Ayano, Mitsui Hinako, Yamaguchi Yohei, Hisada Tomoka, Toyama Tatsuya, Ohya Susumu

Enhancing CYP3A4 Inhibition Prediction Using a Hybrid GNN-ML Model with Data Augmentation

利用数据增强的混合 GNN-ML 模型提高 CYP3A4 抑制预测的准确性

Woo, Somin; Jeon, Ju-Hyeok; Han, Sangil; Lee, Changkyu; Min, Sang-Hyun

Case Report: Pediatric isavuconazole supratherapeutic exposure: a case of long-term use, CYP3A5 poor metabolizer genotype and concomitant CYP3A4 medications

病例报告:儿童异沙康唑超治疗剂量暴露:一例长期用药、CYP3A5代谢能力弱基因型及同时服用CYP3A4药物的病例

Liu, Manman; Li, Lan; Zhou, Chen; Luo, Changying; Wang, Xiaodong; Wu, Juan

Lipid Dependence of CYP3A4 Activity in Nanodiscs

纳米盘中CYP3A4活性的脂质依赖性

Denisov, Ilia G; Grinkova, Yelena V; Sligar, Stephen G

TNFAIP1 suppresses hepatocellular carcinoma progression via the PXR/CYP3A4 signaling axis

TNFAIP1通过PXR/CYP3A4信号通路抑制肝细胞癌的进展。

Nie, Qian; Guo, Yiping; Xiao, Haowen; Zhang, Dini; Li, Haiyue; Wang, Ling

Evaluation of Drug-Drug Interaction Potential Between the Oral Antibiotic Zoliflodacin and the CYP3A4 Inhibitor Itraconazole: A Phase 1 Study in Healthy Participants

口服抗生素佐利氟达星与CYP3A4抑制剂伊曲康唑药物相互作用潜力的评估:一项针对健康受试者的1期研究

Luckey, Alison; Larson, Kajal B; Rayad, Noha; Heep, Markus; Delhomme, Sophie; Kornmann, Gabrielle; Mueller, John P; O'Donnell, John P; O'Brien, Seamus; Fuhr, Rainard; Gillon, Jean-Yves

Dexamethasone-Mediated Regulation of CYP3A4 and UGTs in Human Hepatoma HuH-7 Cells

地塞米松介导的人肝癌HuH-7细胞中CYP3A4和UGT的调控

Yu, Hana; Lee, Song Hee; Kim, Ji Hyeon; Kim, Seung Jin; Kang, Hee Eun

"Reconsidering CYP3A4/5 Genotyping for Ticagrelor Safety: Critical Appraisal of a Narrow Genetic Framework"

“重新审视CYP3A4/5基因分型在替格瑞洛安全性评估中的应用:对狭义遗传框架的批判性评价”

Tahir, Ibadullah; Shahbaz, Hunain