日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

PHI-501, a dual inhibitor of RAF and DDR1/2, overcomes MAPK drug resistance in Melanoma

PHI-501 是一种 RAF 和 DDR1/2 双重抑制剂,可克服黑色素瘤中的 MAPK 药物耐药性。

Kim, Sue Min; Cho, Sungmin; Sung, Gi-Jun; Nam, Ky-Youb; Yoon, JeongHyeok; Sim, Taebo; Ahn, Joong Bae; Shin, Sang Joon

DDR1 Regulates Femoral Arterial Calcification in Lower-Extremity Artery Disease Through NF-Kappa B Activation.

DDR1 通过 NF-κB 激活调节下肢动脉疾病中的股动脉钙化。

Thakur Manovriti, Quillard Thibaut, Angliker Nico, Siegrist Mark, Jansen Yvonne, Yan Yi, Wollenhaupt Julia, Goettsch Claudia, Maegdefessel Lars, Sachs Nadia, Schindewolf Marc, Kotelis Drosos, Noels Heidi, Döring Yvonne

Evaluation of Discoidin domain receptor 1 (DDR1) in junctional epithelial permeability and wound healing.

评估盘状结构域受体 1 (DDR1) 在连接上皮通透性和伤口愈合中的作用。

Zachariadou Christina, Doshi Anuja, Tatakis Dimitris N, Foster Brian L

RAF1 as a standalone therapeutic target in KRAS-driven lung adenocarcinoma: No added efficacy from co-targeting ARAF, EGFR, or DDR1

RAF1 作为 KRAS 驱动的肺腺癌的独立治疗靶点:联合靶向 ARAF、EGFR 或 DDR1 并无额外疗效

de-la-Puente-Ovejero, Laura; Fernández-Rodríguez, Ana; Francoz, Sarah; Aizpurua, Gonzalo; Lomba-Riego, Lucía; Drosten, Matthias; Guerra, Carmen; Musteanu, Mónica; Barbacid, Mariano; García-Alonso, Sara

Inflammatory memory disables a DDR1 degradation checkpoint to enable pancreatic cancer growth

炎症性记忆会禁用DDR1内存退化检查点,从而促进胰腺癌的生长。

Yang, Fei; Lin, Bo; Yuan, Zihang; Yuan, Yongkang; Pu, Xiaohong; Wang, Chunlan; Watari, Kosuke; Luo, Rongkui; Sun, Beicheng; Karin, Michael; Su, Hua

Author Correction: Collagenolysis-dependent DDR1 signalling dictates pancreatic cancer outcome

作者更正:胶原溶解依赖性DDR1信号通路决定胰腺癌预后

Su, Hua; Yang, Fei; Fu, Rao; Trinh, Brittney; Sun, Nina; Liu, Junlai; Kumar, Avi; Baglieri, Jacopo; Siruno, Jeremy; Le, Michelle; Li, Yuhan; Dozier, Stephen; Nair, Ajay; Filliol, Aveline; Sinchai, Nachanok; Rosenthal, Sara Brin; Santini, Jennifer; Metallo, Christian M; Molina, Anthony; Schwabe, Robert F; Lowy, Andrew M; Brenner, David A; Sun, Beicheng; Karin, Michael

Collagen Signaling via DDR1 Exacerbates Barriers to Macromolecular Drug Delivery in a 3D Model of Pancreatic Cancer Fibrosis.

DDR1介导的胶原蛋白信号传导加剧了胰腺癌纤维化3D模型中大分子药物递送的障碍。

Ohira Mayu, Kitamura Moe, Iwasaki Hiroyo, Ohta-Okano Haruko, Tsujii Hiyori, Nakamura Reika, Nakazawa Takuya, Nishiguchi Akihiro, Yamamoto Masaya, Osada Kensuke, Toyooka Shinichi, Cabral Horacio, Masamune Atsushi, Kano Mitsunobu R, Tanaka Hiroyoshi Y

Drug screening in 3D microtumors reveals DDR1/2-MAPK12-GLI1 as a vulnerability in cancer-associated fibroblasts.

在 3D 微肿瘤中进行药物筛选发现 DDR1/2-MAPK12-GLI1 是癌症相关成纤维细胞的脆弱性。

Inhibition of DDR1 potentiates carbon ion radiotherapy by promoting ferroptosis and immunogenic death in head and neck squamous cell carcinoma

抑制DDR1可通过促进头颈部鳞状细胞癌中的铁死亡和免疫原性死亡来增强碳离子放射疗法的疗效。

Hu, Wei; Huang, Qingting; Chen, Li; Geng, Shikai; Zhang, Haojiong; Chen, Huaiyuan; Liu, Xingyu; Zhong, Jingqin; Su, Fengtao; Shao, Chunlin; Kong, Lin

Targeted DDR1 Treatment Strategy Enhances PD-1 Immunotherapy Efficacy against Gastric Cancer

靶向DDR1治疗策略可增强PD-1免疫疗法对胃癌的疗效

Tian, Yonggang; Wang, Jun; Qin, Long; Wang, Xiang; Yu, Yi; Sun, Hui; Bai, Feihu; Zhang, Dekui