日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

BMX inhibition overcomes small cell lung cancer chemoresistance by stabilizing E2F1 via ERK1/2-Cyclin D1/CDK4/6 axis.

BMX抑制剂通过ERK1/2-Cyclin D1/CDK4/6轴稳定E2F1,从而克服小细胞肺癌的化疗耐药性。

Wu Ting, Qi Shuang, Shi Chenliang, Wu Chao, Liu Qingwang, Hu Chen, Hu Jie, Wang Aoli, Liu Jing, Qi Ziping, Wang Wenchao, Liu Qingsong

TP53BP2 Promotes Placental Autophagy and Preeclampsia via G9a and DNMT1 Cooperatively Modulating E2F1.

TP53BP2 通过 G9a 和 DNMT1 协同调节 E2F1 促进胎盘自噬和先兆子痫。

E2F1 K117 methylation by SETD6 disrupts BRD4-E2F1 binding and modulates E2F1 chromatin binding and gene regulation in prostate cancer cells.

SETD6 对 E2F1 K117 的甲基化会破坏 BRD4-E2F1 的结合,并调节前列腺癌细胞中 E2F1 的染色质结合和基因调控。

Ulu Gizem Tugce, Kublanovsky Margarita, Shalev Raz, Biton Tzofit Elbaz, Feldman Michal, Murr Sophia, Brockmeyer Jens, Dorscht Franziska, Weirich Sara, Levy Dan, Jeltsch Albert

Druggable target ATAD2 enhances the malignant progression and cooperates with E2F1 to up-regulate PDK1 expression in glioma.

可成药靶点ATAD2增强恶性进展,并与E2F1协同作用上调胶质瘤中的PDK1表达。

BAP1-mediated stabilization of SUFU enhances E2F1 activity and promotes colorectal tumorigenesis

BAP1介导的SUFU稳定作用增强E2F1活性并促进结直肠肿瘤发生

Zhang, Jujin; Li, Kai; Wang, Changan; Kong, Deyu; Liang, Bin; Han, Lili; Liu, Biao; Wang, Kunpeng; Wang, Pengfei; Zhao, Yun; Ma, Liya; Peng, Jiayin

RB1-I680T mutation potentiates tumor growth and chemotherapy sensitivity in non-small cell lung cancer via derepressing E2F1 transcription.

RB1-I680T 突变通过解除 E2F1 转录的抑制,增强非小细胞肺癌的肿瘤生长和化疗敏感性。

Zhu Yilin, Gao Fengyuan, Liu Yu, Wang Jinfu, Liu Fanrong, Wang Biao, Wu Boxuan, Wang Yue, Zhang Yifan, Tian Zhongxian, Mu Ning, Zhang Xianglin, Zhao Xiaogang, Zhao Yunpeng, Li Peichao

CDK4/6i reverse PARPi resistance by targeting the E2F1- MCM2/5 pathway

CDK4/6抑制剂通过靶向E2F1-MCM2/5通路逆转PARP抑制剂耐药性

Feng, Yujie; Fu, Miao; Zheng, Bowen; Lou, Fanzhuoran; Huang, Xintian; Xie, Xiaowen; Tan, Weijuan; Chen, Quan; Zhang, Wenqing; Hong, Yongxiang; Rong, Kaiyi; Shi, Huibo; Hu, Tianhui; Xiao, Li

Cuproptosis-associated PDHA1 promotes sarcoma progression and immunotherapy responsiveness via the E2F1-PD-L1 axis: a multi-omics and clinical validation study

铜凋亡相关PDHA1通过E2F1-PD-L1轴促进肉瘤进展和免疫治疗反应:一项多组学和临床验证研究

Qin, Haotian; Qi, Tiantian; Yao, Nan; Sheng, Weibei; Deng, Jinhao; Qian, Junyu; Wang, Deli; Zeng, Hui; Weng, Jian; Yang, Jun; Yu, Fei

Hyaluronan Ameliorates Viral Pneumonia in Mice and Humans by Inhibiting Transcription Factor E2F1

透明质酸通过抑制转录因子E2F1改善小鼠和人类的病毒性肺炎

Stober, Vandy P; Trempus, Carol S; Galdi, Flavia; Martin, Negin P; Gladwell, Wesley; Cronce, Michael; Cox, Jeffery S; Keasling, Jay D; Budzik, Jonathan; Chen, Shih-Heng; Sakamachi, Yosuke; Li, Jian-Liang; McGee, Christopher A; Zaccaro, Daniel J; Der, Jane S; Tucker, Charles J; Scappini, Erica; Campos Gomez, Javier; Rowe, Steven M; Cowman, Mary K; Barkauskas, Christina E; Lee, Patty J; Markovetz, Matthew R; Button, Brian; Hill, David B; Erxleben, Dorothea A; Hall, Adam R; Liu, Jian; Xu, Yongmei; Pedone, Claudio; Antonelli Incalzi, Raffaele; Matalon, Sadis; Savani, Rashmin C; Garantziotis, Stavros

Distinct Regulation of the ARF and TAp73 Tumor Suppressor Genes by the Transcription Factor E2F1 Enables Discrimination of Cancer Cells from Normal Growing Cells

转录因子E2F1对ARF和TAp73肿瘤抑制基因的独特调控作用,使得区分癌细胞和正常生长细胞成为可能。

Zhou, Yaxuan; Nakajima, Rinka; Shirasawa, Mashiro; Fikriyanti, Mariana; Watanabe, Ako; Yang, Caiwei; Iwanaga, Ritsuko; Bradford, Andrew P; Kurayoshi, Kenta; Araki, Keigo; Ohtani, Kiyoshi