IL3RA-Targeting Antibody-Drug Conjugate BAY-943 with a Kinesin Spindle Protein Inhibitor Payload Shows Efficacy in Preclinical Models of Hematologic Malignancies
靶向IL3RA的抗体药物偶联物BAY-943,携带驱动蛋白纺锤体蛋白抑制剂有效载荷,在血液系统恶性肿瘤的临床前模型中显示出疗效。
期刊:Cancers
影响因子:4.4
doi:10.3390/cancers12113464
Kirchhoff, Dennis; Stelte-Ludwig, Beatrix; Lerchen, Hans-Georg; Wengner, Antje Margret; Ahsen, Oliver von; Buchmann, Pascale; Märsch, Stephan; Mahlert, Christoph; Greven, Simone; Dietz, Lisa; Erkelenz, Michael; Zierz, Ruprecht; Johanssen, Sandra; Mumberg, Dominik; Sommer, Anette